Cs(2)CO(3)-N,N-Dimethylacetamide-Promoted Esterification of Arylformic Acids with a-Bromo Esters via Nucleophilic Substitution

Cs(2)CO(3)-N,N-二甲基乙酰胺促进芳基甲酸与α-溴代酯的亲核取代酯化反应

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Abstract

Herein, a nucleophilic substitution reaction between arylformic acids and α-bromo esters, facilitated by a Cs(2)CO(3)-DMA system, is reported. This reaction occurs under mild conditions, yielding a diverse range of valuable lactic acid derivatives (34 examples) with good to excellent yields (up to 97%). Subtle factors, such as the ion-dipole interactions between Cs(2)CO(3), the substrates, and the solvent, may significantly influence the dynamics of the S(N)2 reaction.

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