Journal of Combinatorial Chemistry

Design, synthesis, and in vitro evaluation of potential West Nile virus protease inhibitors based on the 1-oxo-1,2,3,4-tetrahydroisoquinoline and 1-oxo-1,2-dihydroisoquinoline scaffolds

基于 1-氧代-1,2,3,4-四氢异喹啉和 1-氧代-1,2-二氢异喹啉骨架的潜在西尼罗河病毒蛋白酶抑制剂的设计、合成及体外评估

Dipeptidyl-quinolone derivatives inhibit hypoxia inducible factor-1α prolyl hydroxylases-1, -2, and -3 with altered selectivity

二肽基喹诺酮衍生物以改变的选择性抑制缺氧诱导因子-1α脯氨酰羟化酶-1、-2和-3

Microwave-assisted fluorous synthesis of a 1,4-benzodiazepine-2,5-dione library.

Rapid and efficient hydrophilicity tuning of p53/mdm2 antagonists.

On-bead screening of combinatorial libraries: reduction of nonspecific binding by decreasing surface ligand density

组合文库的珠上筛选：通过降低表面配体密度来减少非特异性结合

Estimating protein-ligand binding affinity using high-throughput screening by NMR

使用 NMR 高通量筛选评估蛋白质-配体结合亲和力

Fluorous mixture synthesis of two libraries with hydantoin-, and benzodiazepinedione-fused heterocyclic scaffolds

含乙内酰脲和苯二氮卓二酮融合杂环骨架的两个化合物库的氟混合物合成

Plate-to-plate fluorous solid-phase extraction for solution-phase parallel synthesis

用于溶液相平行合成的板对板氟固相萃取