Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC)
高效IDO1蛋白水解靶向嵌合体(PROTAC)的合理设计与优化
期刊:J Med Chem
影响因子:6.800
doi:10.1021/acs.jmedchem.5c00026
Paige J Monsen ,Prashant V Bommi ,Arabela A Grigorescu ,Kristen L Lauing ,Yingyu Mao ,Payton Berardi ,Lijie Zhai ,Oluwatomilayo Ojo ,Manon Penco-Campillo ,Taylor Koch ,Michael Egozi ,Sonam Jha ,Sara F Dunne ,Hong Jiang ,Guiqin Song ,Fang Zhang ,Steven Kregel ,Ali Vaziri-Gohar ,Sean W Fanning ,Pilar Sanchez-Gomez ,Jacob M Allen ,Bakhtiar Yamini ,Rimas V Lukas ,Derek A Wainwright ,Gary E Schiltz