Emerging role of Janus kinase inhibitors in ulcerative colitis management

Janus激酶抑制剂在溃疡性结肠炎治疗中的新兴作用

阅读:1

Abstract

Ulcerative colitis (UC) is a chronic inflammatory bowel disease having high morbidity and a significant negative influence on patients' quality of life. Traditional medicinal strategies available, including amino salicylates, corticosteroids, and biologics, offer limited efficacy, safety, and durability of response. The advancement in small-molecule Janus kinase (JAK) inhibitors has introduced a novel, oral therapeutic option that targets intracellular signaling pathways implicated in UC pathogenesis. Tofacitinib is the first approved JAK inhibitor for the treatment of moderate-to-severe UC. This drug, despite offering promising efficacy, has various safety concerns, especially the occurrence of thromboembolic events. These adverse effects have stressed the development of more selective agents such as upadacitinib and filgotinib. This mini-review explores the current perspectives of JAK inhibitors in UC, particularly focusing on their mechanisms of action, safety profiles, clinical trial outcomes, and emerging strategies to enhance their use. This review also highlights future directions, including the potential of selective JAK1 inhibition and the role of personalized medicine in refining therapeutic decisions. Understanding the emerging place of JAK inhibitors within the UC treatment strategies offers excellent opportunities to increase patient care and long-term disease management.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。