Pse-T2-Based Short Peptides with Broad-Spectrum Antimicrobial Activity, Stability, and Safety Combat MDR Staphylococcus aureus In Vitro and in Mouse Infection Model

基于Pse-T2的短肽具有广谱抗菌活性、稳定性和安全性,可在体外和鼠感染模型中对抗耐多药金黄色葡萄球菌。

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Abstract

Infections caused by MDR pathogens are on the rise worldwide, and relying on conventional antibiotics can be life-threatening for patients. To address this issue, we used a functional truncated peptide, Pse-T2-C12, which exhibited excellent antibacterial, antibiofilm, and antipersister activities, along with a rapid killing rate against all tested pathogens. Pse-T2-C12 kills bacterial cells via pore formation, permeabilization, and disruption of bacterial membranes. Pse-T2-C12 did not induce resistance development, remained stable over pH, temperature, and serum conditions, and showed no detectable toxicity in vitro and in vivo. Moreover, in vivo data showed that Pse-T2-C12 reduced MDR Staphylococcus aureus infection, resulting in a reduced inflammatory response, decreased coagulation, and pain reduction. These findings highlight Pse-T2-C12 as a promising antibiotic candidate owing to its easy synthesis, economic benefits, and ability to treat MDR bacterial infections.

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