Luminescent Assay for the Screening of SARS-CoV-2 M(Pro) Inhibitors

用于筛选SARS-CoV-2 M(Pro)抑制剂的发光检测法

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Abstract

Since the outbreak of SARS-CoV-2 in December 2019 millions of infections have been reported globally. The viral chymotrypsin-like main protease (M(Pro) ) exhibits a crucial role in viral replication and represents a relevant target for antiviral drug development. In order to screen potential M(Pro) inhibitors we developed a luminescent assay using a peptide based probe containing a cleavage site specific for M(Pro) . This assay was validated showing IC(50) values similar to those reported in the literature for known M(Pro) inhibitors and can be used to screen new inhibitors.

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