Preclinical and Case Series Studies on the Combination of Venetoclax with Epigenetic Drugs in T-Cell Acute Lymphoblastic Leukemia

维奈托克联合表观遗传药物治疗T细胞急性淋巴细胞白血病的临床前研究和病例系列研究

阅读:1

Abstract

Adult T-cell acute lymphoblastic leukemia (T-ALL) exhibits a dismal prognosis characterized by low remission rates, high relapse rates, and poor tolerance to conventional chemotherapy. The urgent development of novel therapeutic strategies is imperative to improve clinical outcomes. In this study, we propose a dual epigenetic targeting regimen combining Venetoclax with Chidamide and Azacitidine. Preclinical investigations demonstrated synergistic anti-proliferative effects of this triple-drug combination against Jurkat cells in vitro. Additionally, we retrospectively analyzed clinical data from five high-risk T-ALL patients to evaluate the regimen's efficacy and safety. Among the cohort (all male; median age 55 years, range 25-72), one patient had refractory T-ALL (R-TALL) following VDCP regimen induction failure, while four were newly diagnosed (ND-TALL). After one treatment cycle, four patients achieved complete remission (CR) or CR with incomplete hematologic recovery (CRi), with one additional patient attaining CR after the second cycle. Four patients achieved deep molecular remission (MRD-negative status) within two cycles, while two successfully underwent allogeneic hematopoietic stem cell transplantation (HSCT) during sustained remission. Myelosuppression emerged as the predominant treatment-related adverse event. These preclinical and clinical findings collectively support the therapeutic potential of the Combination of Venetoclax with Epigenetic Drugs as a promising option for high-risk T-ALL patients.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。