Network pharmacology, molecular docking, and dynamics reveal the mechanisms of Hejie Shengfa Decoction against alopecia areata

网络药理学、分子对接和动力学揭示了合节生发汤治疗斑秃的机制

阅读:2

Abstract

Alopecia areata (AA) is a non-scarring autoimmune disorder characterized by patchy hair loss. Hejie Shengfa Decoction (HSD), a Traditional Chinese Medicine formula, has shown clinical efficacy in treating AA, but its molecular mechanisms remain unclear. In this study, network pharmacology, molecular docking, and molecular dynamics simulations were used to explore the potential mechanisms of HSD in AA treatment. Active compounds and their corresponding targets were identified from the Traditional Chinese Medicine Systems Pharmacology Database and Analysis Platform and HERB databases, while AA-related targets were retrieved from GeneCards, OMIM, DrugBank, and DisGeNET. STRING and Cytoscape software were used to construct a protein-protein interaction network. A total of 95 overlapping targets were identified, with core targets including IL6, EGFR, ALB, CASP3, and GAPDH. Gene ontology enrichment analysis revealed that these targets are primarily involved in immune regulation, oxidative stress, and apoptosis. Kyoto Encyclopedia of Genes and Genomes pathway analysis highlighted significant enrichment in the AGE-RAGE, TNF, PI3K-Akt, and JAK-STAT signaling pathways. Molecular docking demonstrated strong binding affinity between stigmasterol and EGFR (-8.3 kcal/mol), which was further validated by molecular dynamics simulations. These findings suggest that HSD may exert therapeutic effects against AA by modulating immune and inflammatory signaling pathways, regulating apoptosis, and improving the follicular microenvironment. This study provides a theoretical foundation for the development of HSD as a natural therapeutic agent for alopecia areata.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。