Kinetic Study of CO(2) Hydration by Small-Molecule Catalysts with A Second Coordination Sphere that Mimic the Effect of the Thr-199 Residue of Carbonic Anhydrase

利用具有第二配位层的小分子催化剂模拟碳酸酐酶Thr-199残基的作用,研究CO₂水合反应的动力学

阅读:1

Abstract

Zinc complexes were synthesized as catalysts that mimic the ability of carbonic anhydrase (CA) for the CO(2) hydration reaction (H(2)O + CO(2) → H(+) + HCO(3)(-)). For these complexes, a tris(2-pyridylmethyl)amine (TPA) ligand mimicking only the active site, and a 6-((bis(pyridin-2-ylmethyl)amino)methyl)pyridin-2-ol (TPA-OH) ligand mimicking the hydrogen-bonding network of the secondary coordination sphere of CA were used. Potentiometric pH titration was used to determine the deprotonation ability of the Zn complexes, and their pK(a) values were found to be 8.0 and 6.8, respectively. Stopped-flow spectrophotometry was used to confirm the CO(2) hydration rate. The rate constants were measured to be 648.4 and 730.6 M(-1)s(-1), respectively. The low pK(a) value was attributed to the hydrogen-bonding network of the secondary coordination sphere of the catalyst that mimics the behavior of CA, and this was found to increase the CO(2) hydration rate of the catalyst.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。