Isoprenylated Flavonoids as Ca(v)3.1 Low Voltage-Gated Ca(2+) Channel Inhibitors from Salvia digitaloides

异戊二烯化黄酮类化合物作为鼠尾草中Ca(v)3.1低电压门控Ca(2+)通道抑制剂

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Abstract

Saldigones A-C (1, 3, 4), three new isoprenylated flavonoids with diverse flavanone, pterocarpan, and isoflavanone architectures, were characterized from the roots of Salvia digitaloides, together with a known isoprenylated flavanone (2). Notably, it's the first report of isoprenylated flavonoids from Salvia species. The structures of these isolates were elucidated by extensive spectroscopic analysis. All of the compounds were evaluated for their activities on Ca(v)3.1 low voltage-gated Ca(2+) channel (LVGCC), of which 2 strongly and dose-dependently inhibited Ca(v)3.1 peak current.

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