A tripartite therapeutic agent reprograms the myocardial infarction microenvironment

三元治疗剂可重塑心肌梗死微环境

阅读:2

Abstract

Myocardial infarction (MI) remains a global health challenge despite advances in reperfusion therapies, as subsequent oxidative stress, inflammatory cascades, and electrical conduction abnormalities impede functional recovery. This study presents a tripartite therapeutic strategy addressing these pathological mechanisms through a clinically translatable multifunctional myocardial repair agent (MMRA). The system combines polypyrrole's and sinomenine's (Sino) anti-inflammatory/antioxidant effects, formulated within a conductive thermoresponsive Poloxamer 407 (P407) hydrogel platform. Injectable P407 hydrogel facilitates targeted delivery and sustained release of therapeutic components within the infarct zone. In vivo evaluations revealed MMRA's capacity to simultaneously: 1) Scavenge reactive oxygen species and downregulate pro-inflammatory cytokines, 2) Reprogram macrophage polarization toward tissue-reparative M2 phenotypes and 3) Restore electrical signal propagation through conductive hydrogel-mediated intercellular coupling. By synergistically modulating the post-infarction microenvironment while preserving myocardial electromechanical synchronization, this integrated therapeutic paradigm demonstrates significant potential for enhancing cardiac repair outcomes. The employment of clinically approved components (Sino and P407) further shows the excellent translational feasibility of the MMRA for MI treatment.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。