TRIP13 alters mitochondrial function and promotes bortezomib resistance in multiple myeloma

TRIP13 改变线粒体功能并促进多发性骨髓瘤对硼替佐米的耐药性

阅读:4

Abstract

Bortezomib (BTZ) resistance remains a major therapeutic challenge in multiple myeloma (MM). This study investigates the role of thyroid hormone receptor interactor 13 (TRIP13) in MM progression and BTZ resistance. Analysis of public datasets and clinical bone marrow samples revealed that TRIP13 is significantly upregulated in MM and that its expression correlates with advanced disease stage and poor overall survival. In vitro, TRIP13 overexpression (TRIP13-OE) in MM cell lines significantly enhanced cell proliferation, reduced BTZ-induced apoptosis, and alleviated G2/M cell cycle arrest. Functional assays further showed that TRIP13-OE cells preserved mitochondrial membrane potential, reduced mitochondrial calcium overload, and maintained ATP production following BTZ exposure. Quantitative polymerase chain reaction (qPCR) analysis demonstrated that mitochondrial regulatory genes were upregulated in TRIP13-OE cells, particularly mitochondrial calcium uniporter (MCU). Co-immunoprecipitation following BTZ treatment confirmed a specific interaction between TRIP13 and MCU, while immunofluorescence labeling showed their cytoplasmic co-localization. These findings uncover a previously unrecognized role of TRIP13 in regulating mitochondrial integrity under proteotoxic stress, thereby contributing to BTZ resistance. Targeting TRIP13 may represent a novel therapeutic approach to improve outcomes in MM patients.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。