In vitro characterisation of fluticasone propionate and ciclesonide delivered with and without valved holding chambers using cascade impaction and an adult simulated breathing profile

采用级联冲击法和模拟成人呼吸模式,对有无阀门储液罐给药的丙酸氟替卡松和环索奈德进行体外表征。

阅读:2

Abstract

BACKGROUND: Valved holding chambers (VHCs) are not interchangeable. Because VHC design and formulation type influence aerosol behaviour, each VHC-drug combination should be evaluated to inform clinical use and device selection. AIM: To compare the aerodynamic particle size distribution (APSD) of two inhaled corticosteroids delivered from pressurised metered dose inhalers with and without commonly used VHCs under realistic, adult-representative breathing. METHODS: We assessed fluticasone propionate (FP, suspension) and ciclesonide (CIC, solution) using no VHC and three VHCs (AeroChamber, EasyChamber and OptiChamber Diamond). A Next Generation Impactor was connected to an anatomically representative adult throat model and a breathing simulator generating an adult-type inhalation profile. RESULTS: Without a VHC, throat deposition was high. With any VHC, throat deposition fell to only a few per cent of the label claim for both FP and CIC. The 1-5 µm respirable fraction was approximately one-third of the label claim for both drugs, irrespective of VHC use, while CIC generated a larger submicron fraction than FP. Small statistically significant differences between VHCs were observed, but absolute differences in APSD and throat deposition were modest. CONCLUSIONS: In adult-representative conditions, VHCs substantially reduce oropharyngeal deposition but do not influence fine-particle delivery. Differences between the tested VHCs were minor and unlikely to be clinically meaningful, whereas FP and CIC showed distinct APSD profiles consistent with formulation type. These findings support performance-based, drug-specific evaluation of VHCs and underscore the value of systematic in vitro testing to guide evidence-based spacer-drug selection and to reduce throat deposition in clinical practice.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。