Neuroprotective potential of polyherbal formulation: Evidence from preliminary in-vitro and in-vivo studies

复方草药制剂的神经保护潜力:来自初步体外和体内研究的证据

阅读:1

Abstract

The objective of the study is to develop and evaluate a polyherbal formulation (PHF) for Parkinson's disease (PD). The present research provides preliminary studies which includes exhaustive literature survey leading to the selection of seven medicinal plants. Hydroalcoholic extracts of these plants were subsequently evaluated for their efficacy using haloperidol catalepsy and antioxidant assay. Based on results, four potent extracts, Asparagus racemosus, Convolvulus prostratus, Bacopa monnieri, and Nigella sativa, were chosen for further research. A PHF containing the above extracts was prepared and assessed for physicochemical properties, microbial load, and bioactive constituents. HPTLC analysis confirmed the presence of quercetin, kaempferol, rutin, and β-sitosterol. Molecular docking was performed for the promising actives present in the above extracts, such as kaempferol, quercetin, rutin, and β-sitosterol, highlighting their potential interactions with the PD-related targets. Antioxidant activity was evaluated using DPPH, ABTS, and FRAP assays, confirming potent free radical scavenging properties. Anti-inflammatory effects were demonstrated via heat-induced hemolysis, albumin denaturation, and proteinase inhibition assays. Additionally, the MAO-B enzyme inhibition assay indicated significant antiparkinsonian potential. PHF, combined with antioxidant, anti-inflammatory, and MAO-B inhibitory activities, supports its therapeutic application in neuronal protection. Acute oral toxicity was assessed as per OECD 425 guidelines, confirming its safety.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。