Bedaquiline Eliminates Bactericidal Activity of β-Lactams against Mycobacterium abscessus

贝达喹啉可消除β-内酰胺类抗生素对脓肿分枝杆菌的杀菌活性

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Abstract

The β-lactams imipenem and cefoxitin are used for the treatment of Mycobacterium abscessus lung infections. Here, we show that these cell wall synthesis inhibitors trigger a lethal bacterial ATP burst by increasing oxidative phosphorylation. Cotreatment of M. abscessus with the antimycobacterial ATP synthase inhibitor bedaquiline suppresses this ATP burst and eliminates the bactericidal activity of β-lactams. Thus, the addition of bedaquiline to β-lactam-containing regimes may negatively affect treatment outcome.

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