Protocol to discover actionable cancer vulnerabilities enabled by neomorph protein-protein interactions with the AVERON Notebook

利用AVERON Notebook发现由新形态蛋白-蛋白相互作用引发的可操作癌症脆弱性的方案

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Abstract

While some tumor driver mutations inhibit existing protein-protein interactions (PPIs), others can create neomorph interactions (neoPPIs) not characteristic of the wild-type counterparts. Such tumor-specific neoPPIs may represent targets for therapeutic interventions. Here, we present a protocol to computationally uncover neoPPI-enabled druggable tumor dependencies using the AVERON Notebook environment. We describe steps for determining PPI levels, identifying clinically significant neoPPIs, and determining neoPPI-regulated pathways. We then detail procedures for determining neoPPI-regulated therapeutically actionable targets. For complete details on the use and execution of this protocol, please refer to Chen et al.(1).

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