日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery, Structure-Activity Relationship, and Functional Characterization of a Chromenopyrrole Series as Orthosteric Antagonists of GPR84

色烯吡咯系列化合物作为GPR84正构拮抗剂的发现、构效关系及功能表征

Malone, Michael A; Yin, Ruijing; Li, Yueming; Jenkins, Laura; Guseinov, Abdul-Akim; Marsango, Sara; Huggett, Mark; Huggett, Margaret; Boyle, Anna; Morrison, Angus; Tikhonova, Irina G; Milligan, Graeme; Jamieson, Andrew G

Steroid Recognition in Adhesion GPCRs: A Structural and Pharmacological Perspective

粘附 GPCR 中的类固醇识别:结构和药理学视角

Fleming, Bethany; Guseinov, Abdul-Akim; Tikhonova, Irina G; Milligan, Graeme; Perry-Hauser, Nicole A

Mechanism of GPR84 allosteric modulation at a helix 8-proximate site

GPR84 在螺旋 8 近端位点的变构调节机制

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Zhou, Jingkai; Gossen, Fabian; Wang, Pinqi; Al Mahmud, Zobaer; Li, Yueming; Mahardhika, Andhika B; Muller, Christa E; Feng, Mingye; Russell, Angela J; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

Allosteric modulation and biased signalling at free fatty acid receptor 2

游离脂肪酸受体 2 的变构调节和偏向性信号传导

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Valentini, Alice; Marsango, Sara; Schultz-Knudsen, Katrine; Ulven, Trond; Rexen Ulven, Elisabeth; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

Steric control of signaling bias in the immunometabolic receptor GPR84

免疫代谢受体 GPR84 中信号偏向的空间控制

Wang, Pinqi; Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; von Hallerstein, Carl; Colburn, Jonathan D; Ives, Rowan; Luscombe, Vincent B; Marsango, Sara; Oktavia, Listiana; Raja, Arun; Greaves, David R; Biggin, Philip C; Milligan, Graeme; Zhang, Cheng; Tikhonova, Irina G; Russell, Angela J

Structural basis for the ligand recognition and signaling of free fatty acid receptors

游离脂肪酸受体的配体识别和信号传导的结构基础

Xuan Zhang, Abdul-Akim Guseinov, Laura Jenkins, Kunpeng Li, Irina G Tikhonova, Graeme Milligan, Cheng Zhang

Exploring an Intracellular Allosteric Site of CC-Chemokine Receptor 4 from 3D Models, Probe Simulations, and Mutagenesis

利用三维模型、探针模拟和诱变技术探索CC趋化因子受体4的细胞内变构位点

Ding, Tianyi; Guseinov, Abdul-Akim; Milligan, Graeme; Plouffe, Bianca; Tikhonova, Irina G

MIS-C related to SARS-CoV-2 infection: a narrative review of presentation, differential diagnosis, and management

与SARS-CoV-2感染相关的MIS-C:临床表现、鉴别诊断和治疗的叙述性综述

Gadiwala, Salika; Mistry, Ayushi; Patel, Sejal; Chaithanya, Avanthika; Pathak, Stuti; Satnarine, Travis; Bekina-Sreenivasan, Daria; Bakarr, Abdul Akim; Das, Bibhuti Bhusan; Chakinala, Raja Chandra; Patel, Saurabhkumar; Areti, Sathya