日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into MERS and SARS coronavirus membrane proteins

对中东呼吸综合征(MERS)和严重急性呼吸综合征(SARS)冠状病毒膜蛋白的结构解析

Mann, Mandeep Kaur; Yin, Yanting; Marsili, Simone; Xie, Jiexiong; Doijen, Jordi; Miller, Robyn; Piassek, Madison; van den Broeck, Nick; Kariuki, Christopher Kinyanjui; de Gruyter, Heidi L M; Leijs, Anouk A; Snijder, Eric J; van Hemert, Martijn J; Keustermans, Ken; Van Gool, Michiel; Yu, Xiaodi; Loock, Marnix van; Koul, Anil; Sharma, Sujata; Van Damme, Ellen; Abeywickrema, Pravien

Discovery of a non-nucleoside inhibitor that binds to a novel site in the palm domain of the respiratory syncytial virus RNA-dependent RNA polymerase.

发现一种非核苷类抑制剂,可与呼吸道合胞病毒 RNA 依赖性 RNA 聚合酶掌状结构域中的新位点结合

Kalin Jay H, Yin Yanting, Tran Minh T, Piassek Madison, Fung Amy, Grosse Sandrine, Jacoby Edgar, Bhaumik Anusarka, Adhikary Suraj, Miller Robyn, Lemmens Cynthia, Lutter Ferdinand H, Pieters Serge, Cooymans Ludwig, Rombouts Geert, Oehlrich Daniel, Tomaso Sonia, Lozada Kate, Garcia Miguel Osorio, Anson Brandon, De Bruyn Suzanne, Smith-Monroy Constance, Neefs Jean-Marc, Conceição-Neto Nádia, Stoops Bart, van Vlijmen Herman, Patrick Aaron, Yu Xiaodi, Wong Victoria, Krosky Daniel, Abeywickrema Pravien, Mason Stephen, Jin Zhinan, Jonckers Tim H M, Sharma Sujata

High-Throughput Assessment of Bile Salt Export Pump Inhibition Using RapidFire-MS and DESI-MS

利用 RapidFire-MS 和 DESI-MS 对胆汁酸输出泵抑制进行高通量评估

Li, Jie; Morato, Nicolás M; Westover, Lori S; Abeywickrema, Pravien; Geng, Jieping; Piassek, Madison; Harden, David; Strambeanu, Iulia; Shi, Zhicai; Cooks, R Graham; Meng, Juncai

Structural understanding of non-nucleoside inhibition in an elongating herpesvirus polymerase.

对延伸疱疹病毒聚合酶中非核苷类抑制剂的结构理解

Hayes Robert P, Heo Mee Ra, Mason Mark, Reid John, Burlein Christine, Armacost Kira A, Tellers David M, Raheem Izzat, Shaw Anthony W, Murray Edward, McKenna Philip M, Abeywickrema Pravien, Sharma Sujata, Soisson Stephen M, Klein Daniel

The methyltransferase domain of the Respiratory Syncytial Virus L protein catalyzes cap N7 and 2'-O-methylation

呼吸道合胞病毒L蛋白的甲基转移酶结构域催化N7帽和2'-O-甲基化。

Sutto-Ortiz, Priscila; Tcherniuk, Sergey; Ysebaert, Nina; Abeywickrema, Pravien; Noël, Mathieu; Decombe, Alice; Debart, Françoise; Vasseur, Jean-Jacques; Canard, Bruno; Roymans, Dirk; Rigaux, Peter; Eléouët, Jean-François; Decroly, Etienne

Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

氨基甲酸酯和N-嘧啶可减轻酰胺水解:基于结构的四氢喹啉IDO1抑制剂药物设计

Li, Derun; Deng, Yongqi; Achab, Abdelghani; Bharathan, Indu; Hopkins, Brett Andrew; Yu, Wensheng; Zhang, Hongjun; Sanyal, Sulagna; Pu, Qinglin; Zhou, Hua; Liu, Kun; Lim, Jongwon; Fradera, Xavier; Lesburg, Charles A; Lammens, Alfred; Martinot, Theodore A; Cohen, Ryan D; Doty, Amy C; Ferguson, Heidi; Nickbarg, Elliott B; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Abeywickrema, Pravien; Andrews, Christine; Chamberlin, Chad; Mabrouk, Omar; Curran, Patrick; Richards, Matthew; Saradjian, Peter; Miller, J Richard; Knemeyer, Ian; Otte, Karin M; Vincent, Stella; Sciammetta, Nunzio; Pasternak, Alexander; Bennett, David Jonathan; Han, Yongxin

Strategic Incorporation of Polarity in Heme-Displacing Inhibitors of Indoleamine-2,3-dioxygenase-1 (IDO1)

策略性地将极性引入血红素置换抑制剂中,以抑制吲哚胺-2,3-双加氧酶-1 (IDO1)

White, Catherine; McGowan, Meredeth A; Zhou, Hua; Sciammetta, Nunzio; Fradera, Xavier; Lim, Jongwon; Joshi, Elizabeth M; Andrews, Christine; Nickbarg, Elliott B; Cowley, Phillip; Trewick, Sarah; Augustin, Martin; von Köenig, Konstanze; Lesburg, Charles A; Otte, Karin; Knemeyer, Ian; Woo, Hyun; Yu, Wensheng; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Curran, Patrick; Heo, Mee Ra; Abeywickrema, Pravien; Miller, J Richard; Bennett, David Jonathan; Han, Yongxin

Structural definition and substrate specificity of the S28 protease family: the crystal structure of human prolylcarboxypeptidase

S28蛋白酶家族的结构定义和底物特异性:人脯氨酰羧肽酶的晶体结构

Soisson, Stephen M; Patel, Sangita B; Abeywickrema, Pravien D; Byrne, Noel J; Diehl, Ronald E; Hall, Dawn L; Ford, Rachael E; Reid, John C; Rickert, Keith W; Shipman, Jennifer M; Sharma, Sujata; Lumb, Kevin J