日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Unpredictable Chronic Mild Stress Upregulates Dopamine Receptor Expression Independent of Fatty Acid-Binding Protein 7 Gene Deletion

不可预测的慢性轻度应激可上调多巴胺受体表达,且与脂肪酸结合蛋白7基因缺失无关

Lu, Huy; Roeder, Nicole; Richardson, Brittany; Hamilton, John; Lagamjis, George; Owada, Yuji; Kagawa, Yoshiteru; Sharma, Abhisheak; Thanos, Panayotis K

Physiologically Based Pharmacokinetic Model for Clinical Translation and Prediction of Drug Interaction of the Major Kratom Alkaloid, Mitragynine

基于生理的药代动力学模型用于临床转化和预测主要克拉托姆生物碱帽柱木碱的药物相互作用。

Chiang, Yi-Hua; Kanumuri, Siva Rama Raju; Berthold, Erin C; Kamble, Shyam H; Gour, Abhishek; Kuntz, Michelle A; Senetra, Alexandria S; Mukhopadhyay, Sushobhan; Lin, Zhoumeng; McCurdy, Christopher R; Sharma, Abhisheak

A chromosome-level Mitragyna parvifolia genome unveils spirooxindole alkaloid diversification and mitraphylline biosynthesis.

染色体水平的帽柱木基因组揭示了螺环吲哚生物碱的多样化和帽柱木碱的生物合成

Laforest Larissa C, Nguyen Tuan-Anh M, Matsumoto Gabriel Oliveira, Ramachandria Pavithra, Chanderbali Andre, Kanumuri Siva Rama Raju, Sharma Abhisheak, McCurdy Christopher R, Dang Thu-Thuy T, Nadakuduti Satya Swathi

Assessing molecular changes underlying isopropylated phenyl phosphate (IPP)-induced larval sensorimotor response deficits in zebrafish

评估异丙基苯基磷酸酯(IPP)诱导的斑马鱼幼体感觉运动反应缺陷的分子机制

Sharma, Sunil; Rojas, Alfredo; Gour, Abhishek; Serradimigni, Rosemaria; Leong, Connor; Sharma, Abhisheak; Dasgupta, Subham

Alkaloid biosynthesis in medicinal crop kratom (Mitragyna speciosa) varies with postharvest, genetic, and seasonal factors

药用作物克拉托姆(Mitragyna speciosa)中的生物碱生物合成受采后处理、遗传和季节因素的影响。

Zhang, Mengzi; Lyndon, Annabella; Kanumuri, Siva Rama Raju; Sharma, Abhisheak; Pearson, Brian J; McCurdy, Christopher R; Chen, Jianjun

Dual Opioid-Neuropeptide FF Small Molecule Ligands Demonstrate Analgesia with Reduced Tolerance Liabilities

双重阿片-神经肽FF小分子配体表现出镇痛作用,且耐受性降低

Mottinelli, Marco; Journigan, V Blair; Obeng, Samuel; Pallares, Victoria L C; Mѐsangeau, Christophe; Kapanda, Coco N; Cutler, Stephen J; Lambert, Janet A; Eans, Shainnel O; Ganno, Michelle L; Sheng, Wanhui; King, Tamara; Sharma, Abhisheak; Mollereau, Catherine; Avery, Bonnie A; McLaughlin, Jay P; McCurdy, Christopher R

DR5 Disulfide Bonding Functions as a Sensor and Effector of Protein Folding Stress

DR5二硫键作为蛋白质折叠应激的传感器和效应器发挥作用

Mary E Law # ,Zaafir M Dulloo # ,Samantha R Eggleston ,Gregory P Takacs ,Grace M Alexandrow ,Young Il Lee ,Mengxiong Wang ,Brian Hardy ,Hanyu Su ,Bianca Forsyth ,Parag Das ,Pran K Datta ,Chi-Wu Chiang ,Abhisheak Sharma ,Siva Rama Raju Kanumuri ,Olga A Guryanova ,Jeffrey K Harrison ,Boaz Tirosh ,Ronald K Castellano ,Brian K Law

Beta-cyclodextrin formulation of a disulfide-bond disrupting agent for improved systemic exposure

β-环糊精制剂的二硫键破坏剂,可提高全身暴露量

Dulloo, Zaafir M; Ghiviriga, Ion; Law, Mary E; Verma, Sarvesh K; Sharma, Abhisheak; Law, Brian K; Castellano, Ronald K

Effects of cannabis smoke and oral Δ9THC on cognition in young adult and aged rats

大麻烟雾和口服Δ9THC对青年和老年大鼠认知能力的影响

Zequeira, Sabrina; Gazarov, Emely A; Güvenli, Alara A; Berthold, Erin C; Senetra, Alexandria S; Febo, Marcelo; Hiranita, Takato; McMahon, Lance R; Sharma, Abhisheak; McCurdy, Christopher R; Setlow, Barry; Bizon, Jennifer L

Discovery of CRBN-recruiting PROTAC degraders of the METTL3-METTL14 complex

发现 CRBN 募集的 METTL3-METTL14 复合物 PROTAC 降解酶

Smith, Alexis R; Nar, Rukiye; Li, Yafang; Gour, Abhishek; Sharma, Abhisheak; Qian, Zhijian; Zheng, Guangrong; Wu, Zhixing