日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A long-lasting PI3Kδ inhibitor zandelisib forms a water-shielded hydrogen bond with p110δ and demonstrates sustained inhibitory effects.

长效 PI3Kδ 抑制剂 zandelisib 与 p110δ 形成水屏蔽氢键,并表现出持续的抑制作用

Kunieda Kana, Nagiri Chisae, Watanabe Miwa, Yoshida Tadashi, Zou Jian, Kaneda Ayumi, Takahashi Yuichi, Aburai Kenichi, Saito Jun-Ichi, Umehara Hiroshi, Otsu Yoshiaki, Ishii Toshihiko

Direct entry of cell-penetrating peptide can be controlled by maneuvering the membrane curvature

通过控制细胞膜曲率可以控制细胞穿透肽的直接进入。

Sakamoto, Kazutami; Morishita, Taku; Aburai, Kenichi; Ito, Daisuke; Imura, Tomohiro; Sakai, Kenichi; Abe, Masahiko; Nakase, Ikuhiko; Futaki, Shiroh; Sakai, Hideki

Key Process and Factors Controlling the Direct Translocation of Cell-Penetrating Peptide through Bio-Membrane

细胞穿透肽直接穿过生物膜的关键过程和控制因素

Sakamoto, Kazutami; Morishita, Taku; Aburai, Kenichi; Sakai, Kenichi; Abe, Masahiko; Nakase, Ikuhiko; Futaki, Shiroh; Sakai, Hideki

Altered sphingoid base profiles predict compromised membrane structure and permeability in atopic dermatitis

鞘氨醇碱基谱的改变预示着特应性皮炎中膜结构和通透性的受损

Loiseau, Nicolas; Obata, Yasuko; Moradian, Sam; Sano, Hiromu; Yoshino, Saeko; Aburai, Kenichi; Takayama, Kozo; Sakamoto, Kazutami; Holleran, Walter M; Elias, Peter M; Uchida, Yoshikazu