日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hydroxamate-based inhibitors reveal structural determinants of selectivity for Plasmodium falciparum aminopeptidase P

基于羟肟酸酯的抑制剂揭示了恶性疟原虫氨肽酶P选择性的结构决定因素

Mills, Belinda J; Gregory, Kyle S; Cozier, Gyles E; Taweechai, Supannee; Loughlan, Eve; McConkey, Glenn A; Isaac, R Elwyn; Foster, Richard; Acharya, K Ravi

Molecular basis of domain-specific angiotensin I-converting enzyme inhibition by the antihypertensive drugs enalaprilat, ramiprilat, trandolaprilat, quinaprilat and perindoprilat

抗高血压药物依那普利拉、雷米普利拉、群多普利拉、喹那普利拉和培哚普利拉对血管紧张素I转化酶的结构域特异性抑制的分子基础

Gregory, Kyle S; Ramasamy, Vinasha; Sturrock, Edward D; Acharya, K Ravi

Design of Novel Mercapto-3-phenylpropanoyl Dipeptides as Dual Angiotensin-Converting Enzyme C-Domain-Selective/Neprilysin Inhibitors.

设计新型巯基-3-苯基丙酰二肽作为双重血管紧张素转换酶C结构域选择性/脑啡肽酶抑制剂

Cozier Gyles E, Coulson Lauren B, Eyermann Charles J, Basarab Gregory S, Schwager Sylva L, Chibale Kelly, Sturrock Edward D, Acharya K Ravi

Molecular Basis of Dipeptide Recognition in Drosophila melanogaster Angiotensin I-Converting Enzyme Homologue, AnCE

果蝇血管紧张素I转化酶同源物(AnCE)中二肽识别的分子基础

Żukowska, Joanna; Gregory, Kyle S; Robinson, Adam; Isaac, R Elwyn; Acharya, K Ravi

Ciprofloxacin Inhibits Angiotensin I‑Converting Enzyme (ACE) Activity by Binding at the Exosite, Distal to the Catalytic Pocket

环丙沙星通过与催化口袋远端的外位点结合来抑制血管紧张素I转化酶(ACE)的活性。

Gregory, Kyle S; Ramasamy, Vinasha; Sturrock, Edward D; Acharya, K Ravi

Molecular basis of acyl-CoA ester recognition by α-methylacyl-CoA racemase from Mycobacterium tuberculosis

结核分枝杆菌α-甲基酰基辅酶A消旋酶识别酰基辅酶A酯的分子基础

Mojanaga, Otsile O; Woodman, Timothy J; Lloyd, Matthew D; Acharya, K Ravi

Correction: Molecular basis of acyl-CoA ester recognition by α-methylacyl-CoA racemase from Mycobacterium tuberculosis

更正:结核分枝杆菌α-甲基酰基辅酶A消旋酶识别酰基辅酶A酯的分子基础

Mojanaga, Otsile O; Woodman, Timothy J; Lloyd, Matthew D; Acharya, K Ravi

Structural basis for inhibition of Mycobacterium tuberculosis α-methylacyl-CoA racemase by 2-arylthiopropanoyl-CoA inhibitor analogs

2-芳基硫代丙酰辅酶A抑制剂类似物抑制结核分枝杆菌α-甲基酰基辅酶A消旋酶的结构基础

Mojanaga, Otsile O; Woodman, Timothy J; Lloyd, Matthew D; Acharya, K Ravi

Molecular basis of human angiotensin-1 converting enzyme inhibition by a series of diprolyl-derived compounds

二丙二酰基衍生物抑制人血管紧张素-1转化酶的分子机制

Gregory, Kyle S; Cozier, Gyles E; Fienberg, Stephen; Chibale, Kelly; Sturrock, Edward D; Acharya, K Ravi

Engineering Plastic Eating Enzymes Using Structural Biology

利用结构生物学工程塑料降解酶

Barclay, Amelia; Acharya, K Ravi