日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

High-affinity, structure-validated and selective macrocyclic peptide tools for chemical biology studies of Huntingtin

用于亨廷顿蛋白化学生物学研究的高亲和力、结构验证和选择性大环肽工具

Fanti, Rebeka; Wolf, Esther; Ikenoue, Tatsuya; Deme, Justin C; Balakrishnan, Swati; Keith, Brandon A; Alteen, Matthew G; Chandrasekaran, Renu; Yadav, Manisha; Bhajiawala, Ritika; Ackloo, Suzanne; Feng, Jia; Pouladi, Mahmoud A; Edwards, Aled M; Wilson, Derek J; Lea, Susan M; Suga, Hiroaki; Harding, Rachel J

CACHE Challenge #3: Targeting the Nsp3 Macrodomain of SARS-CoV-2

CACHE挑战赛#3:靶向SARS-CoV-2的Nsp3宏结构域

Herasymenko, Oleksandra; Silva, Madhushika; Correy, Galen J; Abu-Saleh, Abd Al-Aziz A; Ackloo, Suzanne; Arrowsmith, Cheryl; Ashworth, Alan; Ban, Fuqiang; Beck, Hartmut; Bishop, Kevin P; Bohórquez, Hugo J; Bolotokova, Albina; Breznik, Marko; Chau, Irene; Chen, Yu; Cherkasov, Artem; Dehaen, Wim; Della Corte, Dennis; Denzinger, Katrin; Doering, Niklas P; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Gentile, Francesco; Gibson, Elisa; Gokdemir, Ozan; Gunnarsson, Anders; Günther, Judith; Irwin, John J; Jensen, Jan Halborg; Harding, Rachel J; Hillisch, Alexander; Hoffer, Laurent; Hogner, Anders; Hutchinson, Ashley; Kandwal, Shubhangi; Karlova, Andrea; Koirala, Kushal; Kotelnikov, Sergei; Kozakov, Dima; Lee, Juyong; Lee, Soowon; Lessel, Uta; Liu, Sijie; Liu, Xuefeng; Loppnau, Peter; Meiler, Jens; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Oprea, Tudor I; Paige, Brooks; Pandit, Amit; Park, Keunwan; Poda, Gennady; Protopopov, Mykola V; Pütter, Vera; Ravichandran, Rahul; Rognan, Didier; Rosta, Edina; Sabnis, Yogesh; Scott, Thomas; Seitova, Almagul; Sharma, Purshotam; Sindt, François; Song, Minghu; Steinmann, Casper; Stevens, Rick; Talagayev, Valerij; Tararina, Valentyna V; Tarkhanova, Olga; Tingey, Damon; Trant, John F; Treleaven, Dakota; Tropsha, Alexander; Walters, Patrick; Wells, Jude; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zheng, Shuangjia; Fraser, James S; Schapira, Matthieu

Enantioselective protein affinity selection mass spectrometry (E-ASMS)

对映选择性蛋白质亲和力选择质谱法(E-ASMS)

Wang, Xiaoyun; Sun, Jianxian; Ahmad, Shabbir; Yang, Diwen; Li, Fengling; Chan, U Hang; Zeng, Hong; Simoben, Conrad V; Green, Stuart R; Silva, Madhushika; Houliston, Scott; Dong, Aiping; Bolotokova, Albina; Gibson, Elisa; Kutera, Maria; Ghiabi, Pegah; Kondratov, Ivan; Matviyuk, Tetiana; Chuprina, Alexander; Mavridi, Danai; Lenz, Christopher; Joerger, Andreas C; Brown, Benjamin D; Heath, Richard B; Yue, Wyatt W; Robbie, Lucy K; Beyett, Tyler S; Müller, Susanne; Knapp, Stefan; Owen, Dafydd R; Harding, Rachel; Schapira, Matthieu; Brown, Peter J; Santhakumar, Vijayaratnam; Ackloo, Suzanne; Arrowsmith, Cheryl H; Edwards, Aled M; Peng, Hui; Halabelian, Levon

Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells

强效且选择性的 SETDB1 共价负变构调节剂可降低细胞中的甲基转移酶活性

Mélanie Uguen, Devan J Shell, Madhushika Silva, Yu Deng, Fengling Li, Magdalena M Szewczyk, Ka Yang, Yani Zhao, Michael A Stashko, Jacqueline L Norris-Drouin, Jarod M Waybright, Serap Beldar, Justin M Rectenwald, Angie L Mordant, Thomas S Webb, Laura E Herring, Cheryl H Arrowsmith, Suzanne Ackloo, S

Functionally active modulators targeting the LRRK2 WD40 repeat domain identified by FRASE-bot in CACHE Challenge #1

在 CACHE Challenge #1 中,FRASE-bot 鉴定出了靶向 LRRK2 WD40 重复结构域的功能活性调节因子。

Akhila Mettu,Marta Glavatskikh,Xiaowen Wang,Antonio Jesús Lara Ordóñez,Fengling Li,Irene Chau,Suzanne Ackloo,Cheryl Arrowsmith,Albina Bolotokova,Pegah Ghiabi,Elisa Gibson,Levon Halabelian,Scott Houliston,Rachel J Harding,Ashley Hutchinson,Peter Loppnau,Sumera Perveen,Almagul Seitova,Hong Zeng,Matthieu Schapira,Jean-Marc Taymans,Dmitri Kireev

A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins

WD40重复序列蛋白的靶向配体结合能力评价

Ackloo, Suzanne; Li, Fengling; Szewczyk, Magda; Seitova, Almagul; Loppnau, Peter; Zeng, Hong; Xu, Jin; Ahmad, Shabbir; Arnautova, Yelena A; Baghaie, A J; Beldar, Serap; Bolotokova, Albina; Centrella, Paolo A; Chau, Irene; Clark, Matthew A; Cuozzo, John W; Dehghani-Tafti, Saba; Disch, Jeremy S; Dong, Aiping; Dumas, Antoine; Feng, Jianwen A; Ghiabi, Pegah; Gibson, Elisa; Gilmer, Justin; Goldman, Brian; Green, Stuart R; Guié, Marie-Aude; Guilinger, John P; Harms, Nathan; Herasymenko, Oleksandra; Houliston, Scott; Hutchinson, Ashley; Kearnes, Steven; Keefe, Anthony D; Kimani, Serah W; Kramer, Trevor; Kutera, Maria; Kwak, Haejin A; Lento, Cristina; Li, Yanjun; Liu, Jenny; Loup, Joachim; Machado, Raquel A C; Mulhern, Christopher J; Perveen, Sumera; Righetto, Germanna L; Riley, Patrick; Shrestha, Suman; Sigel, Eric A; Silva, Madhushika; Sintchak, Michael D; Slakman, Belinda L; Taylor, Rhys D; Thompson, James; Torng, Wen; Underkoffler, Carl; von Rechenberg, Moritz; Walsh, Ryan T; Watson, Ian; Wilson, Derek J; Wolf, Esther; Yadav, Manisha; Yazdi, Aliakbar K; Zhang, Junyi; Zhang, Ying; Santhakumar, Vijayaratnam; Edwards, Aled M; Barsyte-Lovejoy, Dalia; Schapira, Matthieu; Brown, Peter J; Halabelian, Levon; Arrowsmith, Cheryl H

OICR-41103 as a chemical probe for the DCAF1 WD40 domain.

OICR-41103 作为 DCAF1 WD40 结构域的化学探针

Kimani Serah W, Noureldin Mahmoud, Wilson Brian, Hoffer Laurent, Green Stuart R, Szewczyk Magdalena M, González-Álvarez Héctor, Mohammed Mohammed, Chan Manuel, Krausser Chiara, Li Alice Shi Ming, Hajian Taraneh, Tucker Sarah, Joshi Dhananjay, Saraon Punit, Thériault Brigitte, Kim Ji Sup, Santhakumar Vijayaratnam, Loppnau Peter, Li Yanjun, Seitova Almagul, Dong Aiping, Kiyota Taira, Hammann Tobias, Gehrtz Paul, Patel Bhashant, Rathod Vaibhavi, Vala Anand, Rout Bhimsen, Jagodra Paras, Brown Peter J, Aman Ahmed, Ramnauth Jailall, Poda Gennady, Uehling David, Arrowsmith Cheryl H, Barsyte-Lovejoy Dalia, Marcellus Richard, Ackloo Suzanne, Mamai Ahmed, Al-Awar Rima, Halabelian Levon

Toward target 2035: EUbOPEN - a public-private partnership to enable & unlock biology in the open

迈向2035年目标:EUbOPEN——一项旨在促进和开放生物学的公私合作项目

Tredup, Claudia; Ackloo, Suzanne; Beck, Hartmut; Brown, Peter J; Bullock, Alex N; Ciulli, Alessio; Dikic, Ivan; Edfeldt, Kristina; Edwards, Aled M; Elkins, Jonathan M; Farin, Henner F; Fon, Edward A; Gstaiger, Matthias; Günther, Judith; Gustavsson, Anna-Lena; Häberle, Sandra; Isigkeit, Laura; Huber, Kilian V M; Kotschy, Andras; Krämer, Oliver; Leach, Andrew R; Marsden, Brian D; Matsui, Hisanori; Merk, Daniel; Montel, Florian; Mulder, Monique P C; Müller, Susanne; Owen, Dafydd R; Proschak, Ewgenij; Röhm, Sandra; Stolz, Alexandra; Sundström, Michael; von Delft, Frank; Willson, Timothy M; Arrowsmith, Cheryl H; Knapp, Stefan

Site-Specific Hydrogen Deuterium Exchange Difference Mass Spectrometry Measurements for Ligand Binding

位点特异性氢氘交换差分质谱测量用于配体结合

Anacleto, Joseph; Ackloo, Suzanne; Arrowsmith, Cheryl; Wolf, Esther; Leblanc, Yves; Lento, Cristina; Wilson, Derek J

Enantioselective Protein Affinity Selection Mass Spectrometry (E-ASMS)

对映选择性蛋白质亲和力选择质谱法 (E-ASMS)

Wang, Xiaoyun; Sun, Jianxian; Ahmad, Shabbir; Yang, Diwen; Li, Fengling; Chan, U Hang; Zeng, Hong; Simoben, Conrad V; Green, Stuart R; Silva, Madhushika; Houliston, Scott; Dong, Aiping; Bolotokova, Albina; Gibson, Elisa; Kutera, Maria; Ghiabi, Pegah; Kondratov, Ivan; Matviyuk, Tetiana; Chuprina, Alexander; Mavridi, Danai; Lenz, Christopher; Joerger, Andreas C; Brown, Benjamin D; Heath, Richard B; Yue, Wyatt W; Robbie, Lucy K; Beyett, Tyler S; Müller, Susanne; Knapp, Stefan; Harding, Rachel; Schapira, Matthieu; Brown, Peter J; Santhakumar, Vijayaratnam; Ackloo, Suzanne; Arrowsmith, Cheryl H; Edwards, Aled M; Peng, Hui; Halabelian, Levon