A reversible allosteric inhibitor of GlyT2 for neuropathic pain without on-target side effects
一种可逆的GlyT2变构抑制剂,用于治疗神经性疼痛,且无靶向副作用。
期刊:Nature Communications
影响因子:15.7
doi:10.1038/s41467-026-69616-5
Cantwell Chater, Ryan P; Peiser-Oliver, Julian; Pati, Tanmay K; Quinn, Ada S; Lotsaris, Irina; Frangos, Zachary J; Anderson, Kristen E; Tischer, Anna E; Williams-Noonan, Billy J; Aubrey, Karin R; O'Mara, Megan L; Michaelides, Michael; Mohammadi, Sarasa A; Cioffi, Christopher L; Vandenberg, Robert J; Shahsavar, Azadeh