日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Efficacy evaluation of the S-adenosylhomocysteine hydrolase inhibitor MSD-914 in rhesus macaques (Macaca Mulatta) challenged with Ebola virus by the intramuscular route

对经肌肉注射途径感染埃博拉病毒的恒河猴(Macaca mulatta)进行S-腺苷高半胱氨酸水解酶抑制剂MSD-914的疗效评价

Johnston, Sara C; Ginnetti, Anthony T; Twenhafel, Nancy A; Norris, Sarah L W; Chen, Shiying; Moore, Josh L; Boyce, Christopher W; Frick, Ondraya M; Dyer, Dave N; Marsh, Donald J; Stevens, Stephen C; Knapp, Walter F; Berrier, Kerry L; Wan, Hui; Adam, Gregory C; Hartingh, Timothy J; Esham, Heather L; Fiallos, Jimmy O; Blue, Eugene L; Sifford, Willie B; Latty, Jonathan D; Mills, Harold L; Alli, Nazira A; Piper, Ashley E; Goodson, Aimee I; Meinig, J Matthew; Olsen, David B; Lieberman, Linda A; Panchal, Rekha G

Fluorinated Isoindolinone-Based Glucosylceramide Synthase Inhibitors with Low Human Dose Projections

基于氟化异吲哚啉酮的葡萄糖基神经酰胺合成酶抑制剂的低剂量人体预测

Loughran, H Marie; Schirripa, Kathy M; Roecker, Anthony J; Breslin, Michael J; Tong, Ling; Fillgrove, Kerry L; Kuo, Yuhsin; Bleasby, Kelly; Collier, Hannah; Altman, Michael D; Ford, Melissa C; Newman, Justin A; Drolet, Robert E; Cosden, Mali; Jinn, Sarah; Flick, Rosemarie B; Liu, Xiaomei; Minnick, Christina; Watt, Marla L; Lemaire, Wei; Burlein, Christine; Adam, Gregory C; Austin, Lauren A; Marcus, Jacob N; Smith, Sean M; Fraley, Mark E

An Application of an Initial Full Value of Vaccine Assessment Methodology to Measles-Rubella MAPs for Use in Low- and Middle-Income Countries

将疫苗初始全面价值评估方法应用于中低收入国家使用的麻疹-风疹微量免疫规划

Ko, Melissa; Frivold, Collrane; Mvundura, Mercy; Soble, Adam; Gregory, Christopher; Christiansen, Hans; Hasso-Agopsowicz, Mateusz; Fu, Han; Jit, Mark; Hsu, Shan; Mistilis, Jessica Joyce; Scarna, Tiziana; Earle, Kristen; Menozzi-Arnaud, Marion; Giersing, Birgitte; Jarrahian, Courtney; Yakubu, Ahmadu; Malvolti, Stefano; Amorij, Jean-Pierre

Pyrazole Ureas as Low Dose, CNS Penetrant Glucosylceramide Synthase Inhibitors for the Treatment of Parkinson's Disease

吡唑脲类药物作为低剂量、可穿透血脑屏障的中枢神经系统葡糖基神经酰胺合成酶抑制剂,用于治疗帕金森病

Roecker, Anthony J; Schirripa, Kathy M; Loughran, H Marie; Tong, Ling; Liang, Tao; Fillgrove, Kerry L; Kuo, Yuhsin; Bleasby, Kelly; Collier, Hannah; Altman, Michael D; Ford, Melissa C; Drolet, Robert E; Cosden, Mali; Jinn, Sarah; Hatcher, Nathan G; Yao, Lihang; Kandebo, Monika; Vardigan, Joshua D; Flick, Rosemarie B; Liu, Xiaomei; Minnick, Christina; Price, Laura A; Watt, Marla L; Lemaire, Wei; Burlein, Christine; Adam, Gregory C; Austin, Lauren A; Marcus, Jacob N; Smith, Sean M; Fraley, Mark E

Improvements to the Gulf pipefish Syngnathus scovelli genome

对墨西哥湾海龙(Syngnathus scovelli)基因组的改进

Ramesh, Balan; Small, Clay M; Healey, Hope; Johnson, Bernadette; Barker, Elyse; Currey, Mark; Bassham, Susan; Myers, Megean; Cresko, William A; Jones, Adam Gregory

SARS-CoV-2 tropism, entry, replication, and propagation: Considerations for drug discovery and development

SARS-CoV-2 的嗜性、入侵、复制和传播:药物发现和开发中的考量

Murgolo, Nicholas; Therien, Alex G; Howell, Bonnie; Klein, Daniel; Koeplinger, Kenneth; Lieberman, Linda A; Adam, Gregory C; Flynn, Jessica; McKenna, Philip; Swaminathan, Gokul; Hazuda, Daria J; Olsen, David B

Redefining the Histone Deacetylase Inhibitor Pharmacophore: High Potency with No Zinc Cofactor Interaction

重新定义组蛋白去乙酰化酶抑制剂药效团:高效且无锌辅因子相互作用

Beshore, Douglas C; Adam, Gregory C; Barnard, Richard J O; Burlein, Christine; Gallicchio, Steven N; Holloway, M Katharine; Krosky, Daniel; Lemaire, Wei; Myers, Robert W; Patel, Sangita; Plotkin, Michael A; Powell, David A; Rada, Vanessa; Cox, Christopher D; Coleman, Paul J; Klein, Daniel J; Wolkenberg, Scott E

Discovery of the First Non-cGMP Mimetic Small Molecule Activators of cGMP-Dependent Protein Kinase 1 α (PKG1α)

发现首个非cGMP模拟小分子cGMP依赖性蛋白激酶1α(PKG1α)激活剂

Hanisak, Jennifer; Soriano, Aileen; Adam, Gregory C; Basso, Andrea; Bauman, David; Bell, David; Frank, Emily; O'Donnell, Gregory; Tawa, Paul; Verras, Andreas; Yu, Yang; Zhang, Lei; Seganish, W Michael