日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of potent and brain-penetrable tubulin inhibitors that effectively suppress breast cancer brain metastasis.

发现强效且能穿透血脑屏障的微管蛋白抑制剂,可有效抑制乳腺癌脑转移。

Krutilina Raisa I, Adeleye Kelli L, Playa Hilaire C, Pochampally Satyanarayana, Banjeree Souvik, Oluwalana Damilola, Kamal Mir Shahriar, Tian Di, Miller Duane D, Li Wei, Seagroves Tiffany N

Biological activity of a stable 6-aryl-2-benzoyl-pyridine colchicine-binding site inhibitor, 60c, in metastatic, triple-negative breast cancer.

稳定的 6-芳基-2-苯甲酰基-吡啶秋水仙碱结合位点抑制剂 60c 在转移性三阴性乳腺癌中的生物活性

Oluwalana Damilola, Adeleye Kelli L, Krutilina Raisa I, Chen Hao, Playa Hilaire, Deng Shanshan, Parke Deanna N, Abernathy John, Middleton Leona, Cullom Alexandra, Thalluri Bhargavi, Ma Dejian, Meibohm Bernd, Miller Duane D, Seagroves Tiffany N, Li Wei