Discovery of Dabrafenib: A Selective Inhibitor of Raf Kinases with Antitumor Activity against B-Raf-Driven Tumors
达拉非尼的发现:一种选择性Raf激酶抑制剂,对B-Raf驱动的肿瘤具有抗肿瘤活性
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/ml4000063
Rheault, Tara R; Stellwagen, John C; Adjabeng, George M; Hornberger, Keith R; Petrov, Kimberly G; Waterson, Alex G; Dickerson, Scott H; Mook, Robert A Jr; Laquerre, Sylvie G; King, Alastair J; Rossanese, Olivia W; Arnone, Marc R; Smitheman, Kimberly N; Kane-Carson, Laurie S; Han, Chao; Moorthy, Ganesh S; Moss, Katherine G; Uehling, David E