日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multiscale-Aware Graph Embedding Approach Uncovers LC-61, a Potent Anti-Leishmania infantum Compound

多尺度感知图嵌入方法揭示了LC-61,一种强效抗婴儿利什曼原虫化合物。

Costa, Vinícius Alexandre Fiaia; Carvalho, Alexandra Maria Dos Santos; Chelucci, Rafael Consolin; Mendonça de Melo, Felipe da Silva; Felizardo, Gustavo Santos Sandes; Bernardes, Clarissa Alves Carneiro; Martin, Holli-Joi; Braga, Rodolpho de Campos; Charneau, Sébastien; Muratov, Eugene N; Andricopulo, Adriano Defini; Bastos, Izabela Marques Dourado; Neves, Bruno Junior

Exploring Bioactive Metabolites From Fusarium falciforme and Aspergillus terreus Isolated From Protease-Rich Fruits: Antifungal, Antitrypanosomal, and Enzymatic Inhibitory Activities

从富含蛋白酶的水果中分离的镰刀菌和土曲霉的生物活性代谢物研究:抗真菌、抗锥虫和酶抑制活性

de Oliveira Almeida, Gabriela; Mazucato, Vitor de Souza; Tonani, Ludmilla; von Zeska Kress, Marcia Regina; Barbosa, Gisele; Krogh, Renata; Andricopulo, Adriano Defini; Gomes Ferreira, Leonardo Luiz; Vieira, Paulo Cezar

Co-cultivation and Medium Optimization: A Strategy for Discovering Fungal-derived Protease Inhibitors

共培养和培养基优化:发现真菌来源蛋白酶抑制剂的策略

Mazucato, Vitor de Souza; Tonani, Ludmilla; von Zeska Kress, Marcia Regina; Andricopulo, Adriano Defini; Barbosa, Gisele; Krogh, Renata; Gomes Ferreira, Leonardo Luiz; Vieira, Paulo Cezar

Optimizing Bothropstoxin-I-Derived Peptides: Exploring the Antibacterial Potential of p-BthW

优化矛头毒素-I 衍生肽:探索 p-BthW 的抗菌潜力

Gabriela Marinho Righetto, Norival Alves Santos-Filho, Letícia Oliveira Catarin Nunes, Camille André, Julia Medeiros Souza, Adriano Defini Andricopulo, Paulo José Martins Bispo, Eduardo Maffud Cilli, Ilana Lopes Baratella da Cunha Camargo

Antimicrobial Activity of an Fmoc-Plantaricin 149 Derivative Peptide against Multidrug-Resistant Bacteria

Fmoc-Plantaricin 149 衍生肽对多药耐药细菌的抗菌活性

Gabriela Marinho Righetto, José Luiz de Souza Lopes, Paulo José Martins Bispo, Camille André, Julia Medeiros Souza, Adriano Defini Andricopulo, Leila Maria Beltramini, Ilana Lopes Baratella da Cunha Camargo

Identification of natural cytochalasins as leads for neglected tropical diseases drug discovery

鉴定天然细胞松弛素作为被忽视的热带疾病药物研发的先导

Marilia Valli, Julia Medeiros Souza, Rafael Consolin Chelucci, Carolina Rabal Biasetto, Angela Regina Araujo, Vanderlan da Silva Bolzani, Adriano Defini Andricopulo

Structure-activity relationships of sulfonamides derived from carvacrol and their potential for the treatment of Alzheimer's disease

香芹酚衍生的磺胺类药物的构效关系及其治疗阿尔茨海默病的潜力

Márcia Maria de Souza, Marina Corrêa Andreolla, Thaís Cecília Ribeiro, Ana Elisa Gonçalves, Alex Rogério Medeiros, Anacleto Silva de Souza, Leonardo Luiz Gomes Ferreira, Adriano Defini Andricopulo, Rosendo Augusto Yunes, Aldo Sena de Oliveira

Novel ruthenium complexes as potential drugs for Chagas's disease: enzyme inhibition and in vitro/in vivo trypanocidal activity

新型钌配合物作为治疗恰加斯病的潜在药物:酶抑制作用及体外/体内锥虫杀灭活性

Silva, Jean Jerley Nogueira; Guedes, Paulo Marcos Matta; Zottis, Aderson; Balliano, Tatiane Luciano; Nascimento Silva, Francisco Ordelei; França Lopes, Luiz Gonzaga; Ellena, Javier; Oliva, Glaucius; Andricopulo, Adriano Defini; Franco, Douglas Wagner; Silva, João Santana