日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multiparameter Kinetic Analysis for Covalent Fragment Optimization by Using Quantitative Irreversible Tethering (qIT)

利用定量不可逆连接(qIT)进行共价片段优化的多参数动力学分析

Craven, Gregory B; Affron, Dominic P; Kösel, Teresa; Wong, Tsz Lam M; Jukes, Zoë H; Liu, Chun-Ting; Morgan, Rhodri M L; Armstrong, Alan; Mann, David J

Vinyl sulfonamide synthesis for irreversible tethering via a novel α-selenoether protection strategy

通过一种新型的α-硒醚保护策略合成用于不可逆连接的乙烯基磺酰胺

Craven, Gregory B; Affron, Dominic P; Raymond, Philip N; Mann, David J; Armstrong, Alan

High-Throughput Kinetic Analysis for Target-Directed Covalent Ligand Discovery

用于靶向共价配体发现的高通量动力学分析

Craven, Gregory B; Affron, Dominic P; Allen, Charlotte E; Matthies, Stefan; Greener, Joe G; Morgan, Rhodri M L; Tate, Edward W; Armstrong, Alan; Mann, David J

Palladium-Catalyzed Directed C(sp(3))-H Arylation of Saturated Heterocycles at C-3 Using a Concise Optimization Approach

利用简洁的优化方法实现钯催化饱和杂环化合物C-3位定向C(sp(3))-H芳基化反应

Affron, Dominic P; Bull, James A

Synthesis and purification of iodoaziridines involving quantitative selection of the optimal stationary phase for chromatography

碘代氮丙啶的合成与纯化,包括色谱法最佳固定相的定量选择

Boultwood, Tom; Affron, Dominic P; Bull, James A