日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Direct-to-Biology Enabled Molecular Glue Discovery

直接应用于生物学领域的分子胶发现

Hu, Maowei; Ochoada, Jason; Actis, Marisa; McGowan, Kevin; Jarusiewicz, Jamie A; Yoshimura, Satoshi; McGrath, Logan; Neelakantan, Uma; Aggarwal, Anup; Mayasundari, Anand; Young, Sarah M; Zhang, Meng; Yang, Lei; Li, Yong; Mercer, Shea; Babu, M Madan; Fischer, Marcus; Young, Brandon M; Yang, Jun J; Nishiguchi, Gisele; Shelat, Anang A; Blair, Daniel J

Unbiased mapping of cereblon neosubstrate landscape by high-throughput proteomics.

利用高通量蛋白质组学对 cereblon 新底物景观进行无偏映射

Steger Martin, Nishiguchi Gisele, Wu Qiong, Schwalb Bjoern, Shashikadze Bachuki, McGowan Kevin, Actis Marisa, Aggarwal Anup, Shi Zhe, Price Jeanine, Mayasundari Anand, Yang Lei, Bednarz Anastasia H, Machata Sophie, Graef Tobias, Bartoschek Denis, Demichev Vadim, Ohmayer Uli, Yang Jun, Daub Henrik, Rankovic Zoran

LCK-targeting molecular glues overcome resistance to inhibitor-based therapy in T-cell acute lymphoblastic leukemia

靶向LCK的分子胶克服了T细胞急性淋巴细胞白血病对抑制剂疗法的耐药性

Yang, Jun J; Nishiguchi, Gisele; Yoshimura, Satoshi; Actis, Marisa; Seffernick, Justin T; Jarusiewicz, Jamie A; Aggarwal, Anup; Li, Angelina; Li, Yong; Lee, DongGeun; Yang, Lei; Mayasundari, Anand; Rankovic, Zoran; Fischer, Marcus

An Antibacterial β-Lactone Kills Mycobacterium tuberculosis by Disrupting Mycolic Acid Biosynthesis

一种抗菌β-内酯通过干扰分枝菌酸生物合成来杀死结核分枝杆菌。

Lehmann, Johannes; Cheng, Tan-Yun; Aggarwal, Anup; Park, Annie S; Zeiler, Evelyn; Raju, Ravikiran M; Akopian, Tatos; Kandror, Olga; Sacchettini, James C; Moody, D Branch; Rubin, Eric J; Sieber, Stephan A