Target deconvolution of HDAC pharmacopoeia reveals MBLAC2 as common off-target
HDAC 药典的靶标反卷积显示 MBLAC2 是常见的脱靶
期刊:Nature Chemical Biology
影响因子:12.9
doi:10.1038/s41589-022-01015-5
Severin Lechner, Martin Ian P Malgapo, Christian Grätz, Raphael R Steimbach, Agnes Baron, Patrick Rüther, Simon Nadal, Carmen Stumpf, Christina Loos, Xin Ku, Polina Prokofeva, Ludwig Lautenbacher, Tino Heimburg, Vivian Würf, Chen Meng, Mathias Wilhelm, Wolfgang Sippl, Karin Kleigrewe, Josch K Paulin