日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

AI Based Discovery of a New AKR1C3 Inhibitor for Anticancer Applications

基于人工智能的新型AKR1C3抑制剂的发现及其在抗癌应用中的应用

Pippione, Agnese C; Vigato, Chiara; Tucciarello, Cristina; Hussain, Samrina; Salladini, Edoardo; Truong, Ha H; Henriksen, Niel M; Vanzetti, Gaia; Giordano, Giorgia; Zonari, Daniele; Mirza, Osman Asghar; Frydenvang, Karla; Pignochino, Ymera; Oliaro-Bosso, Simonetta; Boschi, Donatella; Lolli, Marco L

Exploring the Potential of Sulfur Moieties in Compounds Inhibiting Steroidogenesis

探索硫基团在抑制类固醇生成的化合物中的潜力

Wróbel, Tomasz M; Sharma, Katyayani; Mannella, Iole; Oliaro-Bosso, Simonetta; Nieckarz, Patrycja; Du Toit, Therina; Voegel, Clarissa Daniela; Rojas Velazquez, Maria Natalia; Yakubu, Jibira; Matveeva, Anna; Therkelsen, Søren; Jørgensen, Flemming Steen; Pandey, Amit V; Pippione, Agnese C; Lolli, Marco L; Boschi, Donatella; Björkling, Fredrik

Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5- a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety

使用基于 2-羟基吡唑并 [1,5- a] 吡啶骨架的强效人类二氢乳清酸脱氢酶抑制剂靶向治疗急性髓性白血病:芳氧基芳基部分的 SAR

Stefano Sainas, Marta Giorgis, Paola Circosta, Giulio Poli, Marta Alberti, Alice Passoni, Valentina Gaidano, Agnese C Pippione, Nicoletta Vitale, Davide Bonanni, Barbara Rolando, Alessandro Cignetti, Cristina Ramondetti, Alessia Lanno, Davide M Ferraris, Barbara Canepa, Barbara Buccinnà, Marco Picci

Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5- a]pyridine Scaffold: SAR of the Biphenyl Moiety

使用基于 2-羟基吡唑并 [1,5- a] 吡啶骨架的强效人类二氢乳清酸脱氢酶抑制剂靶向治疗急性髓性白血病:联苯部分的 SAR

Stefano Sainas, Marta Giorgis, Paola Circosta, Valentina Gaidano, Davide Bonanni, Agnese C Pippione, Renzo Bagnati, Alice Passoni, Yaqi Qiu, Carina Florina Cojocaru, Barbara Canepa, Alessandro Bona, Barbara Rolando, Mariia Mishina, Cristina Ramondetti, Barbara Buccinnà, Marco Piccinini, Mohammad Hou

A New NF-κB Inhibitor, MEDS-23, Reduces the Severity of Adverse Post-Ischemic Stroke Outcomes in Rats

新型 NF-κB 抑制剂 MEDS-23 可降低大鼠缺血性卒中后不良后果的严重程度

Rubin, Elina; Pippione, Agnese C; Boyko, Matthew; Einaudi, Giacomo; Sainas, Stefano; Collino, Massimo; Cifani, Carlo; Lolli, Marco L; Abu-Freha, Naim; Kaplanski, Jacob; Boschi, Donatella; Azab, Abed N

N-Acetyl-3-aminopyrazoles block the non-canonical NF-kB cascade by selectively inhibiting NIK

N-乙酰-3-氨基吡唑类化合物通过选择性抑制NIK来阻断非经典NF-κB级联反应。

Pippione, Agnese C; Sainas, Stefano; Federico, Antonella; Lupino, Elisa; Piccinini, Marco; Kubbutat, Michael; Contreras, Jean-Marie; Morice, Christophe; Barge, Alessandro; Ducime, Alex; Boschi, Donatella; Al-Karadaghi, Salam; Lolli, Marco L

4-Hydroxy-N-[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazole-3-carboxamide: a novel inhibitor of the canonical NF-κB cascade

4-羟基-N-[3,5-双(三氟甲基)苯基]-1,2,5-噻二唑-3-甲酰胺:一种新型的经典NF-κB级联抑制剂

Pippione, Agnese C; Federico, Antonella; Ducime, Alex; Sainas, Stefano; Boschi, Donatella; Barge, Alessandro; Lupino, Elisa; Piccinini, Marco; Kubbutat, Michael; Contreras, Jean-Marie; Morice, Christophe; Al-Karadaghi, Salam; Lolli, Marco L

Discovery and verification of panels of T-lymphocyte proteins as biomarkers of Parkinson's disease

发现并验证 T 淋巴细胞蛋白组作为帕金森病的生物标志物

Tiziana Alberio, Agnese C Pippione, Maurizio Zibetti, Simone Olgiati, Daniela Cecconi, Cristoforo Comi, Leonardo Lopiano, Mauro Fasano