日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of cell-active BRD4-D1 selective inhibitors to decode the role of BET proteins in LPS-mediated liver inflammation

开发具有细胞活性的BRD4-D1选择性抑制剂,以揭示BET蛋白在LPS介导的肝脏炎症中的作用

Scholtz, Cole R; Doskey, Luke C; Kandanur, Sai Giridhar Sarma; Vail, Nora R; Roderick, Erika R; Peterson, Elliott J; Hoell, Zachariah J; Shi, Ke; Aihara, Hideki; Kostallari, Enis; Shah, Vijay H; Malhi, Harmeet; Pomerantz, William C K

Structural basis for bat receptor recognition by SARS-CoV-2 and bat SARS2-like coronaviruses

SARS-CoV-2 和蝙蝠 SARS-CoV-2 样冠状病毒识别蝙蝠受体的结构基础

Hsueh, Fu-Chun; Shi, Ke; Aihara, Hideki; Li, Fang

Direct interaction between human DDX1 and SARS-CoV-2 nucleocapsid protein is regulated by phosphorylation

人源DDX1与SARS-CoV-2核衣壳蛋白之间的直接相互作用受磷酸化调控

Wang, Liangjun; Baxley, Ryan M; Largaespada, David A; Aihara, Hideki; Bielinsky, Anja Katrin

The atomic structure of human dystrophin spectrin-like repeat 24

人类肌营养不良蛋白谱蛋白样重复序列24的原子结构

Streeter, Oakley; Shi, Ke; Bui, Hannah; Aihara, Hideki; Ervasti, James M; Evans, Robert 3rd; Muretta, Joseph M

Structural basis for sequence context-independent single-stranded DNA cytosine deamination by the bacterial toxin SsdA.

细菌毒素 SsdA 对单链 DNA 胞嘧啶进行序列上下文无关脱氨的结构基础。

Yin Lulu, Chen Yanjun, Shi Ke, Barreto Duran Emilia, Harris Reuben S, Aihara Hideki

Targeting N-Myc in neuroblastoma with selective Aurora kinase A degraders.

利用选择性 Aurora 激酶 A 降解剂靶向神经母细胞瘤中的 N-Myc

Tang Jian, Moorthy Ramkumar, Hirsch Laura E, Demir Özlem, Baker Zachary D, Naumann Jordan A, Jones Katherine F M, Grillo Michael J, Haefner Ella S, Shi Ke, Levy Michaella J, Gupta Harshita B, Aihara Hideki, Harris Reuben S, Amaro Rommie E, Levinson Nicholas M, Harki Daniel A

Discovery of Small-Molecule Orthopoxvirus Resolvase Inhibitors with Antiviral Activity

发现具有抗病毒活性的小分子正痘病毒分解酶抑制剂

Mahoney, Jacob P; Offei, Samuel; Pant, Anil; Wang, Ziyue; Weiner, Benjamin; Yin, Lulu; Ryu, Won Hee; Katekar, Roshan; Williams, Jessica M; Aihara, Hideki; Yang, Zhilong; Wang, Zhengqiang

Regulatory Interactions between APOBEC3B N- and C-Terminal Domains

APOBEC3B N端和C端结构域之间的调控相互作用

Braza, Mac Kevin E; Demir, Özlem; Ahn, Surl-Hee; Morris, Clare K; Calvó-Tusell, Carla; McGuire, Kelly L; de la Peña Avalos, Bárbara; Carpenter, Michael A; Chen, Yanjun; Casalino, Lorenzo; Aihara, Hideki; Herzik, Mark A Jr; Harris, Reuben S; Amaro, Rommie E

Structural basis for varying drug resistance of SARS-CoV-2 M(pro) E166 variants

SARS-CoV-2 M(pro) E166 变体耐药性差异的结构基础

Esler, Morgan A; Shi, Ke; Rollie, Joseph A; Delgado, Renee; Vishwakarma, Jyoti; Dabrowska, Agnieszka; Prahlad, Janani; Moghadasi, Seyed Arad; Harris, Reuben S; Aihara, Hideki

Human dystrophin tandem calponin homology actin-binding domain crystallized in a closed-state conformation

人类肌营养不良蛋白串联钙调蛋白同源肌动蛋白结合域以闭合状态构象结晶

Streeter, Oakley; Shi, Ke; Vavra, Joseph; Aihara, Hideki; Ervasti, James M; Evans, Robert 3rd; Muretta, Joseph M