日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dendrimer-Conjugated Glutamine Antagonist, D-TTM020, Ameliorates Brain Immune Dysregulation and Improves Neurobehavioral Deficits in the Mecp2-Deficient Mouse Model

树状聚合物偶联的谷氨酰胺拮抗剂D-TTM020可改善Mecp2缺陷小鼠模型的脑免疫失调并改善其神经行为缺陷。

Vyas, Preeti; Khoury, Elizabeth Smith; Sah, Nirnath; Sharma, Anjali; Allende Labastida, Javier; Wilkinson, Elizabeth L; Lac, Kathleen; Damiba, Nerketa N L; Fowler, Amanda; Liu, Jinhuan; Bedner, Ashley; Majer, Pavel; Tichý, Tomás; Thomas, Ajit G; Rais, Rana; Slusher, Barbara S; Kannan, Rangaramanujam M; Kannan, Sujatha

Inhibition of microglial glutaminase alleviates chronic stress-induced neurobehavioral and cognitive deficits

抑制小胶质细胞谷氨酰胺酶可缓解慢性应激引起的神经行为和认知缺陷

Huang, Meixiang; Li, Yannan; Thomas, Ajit G; Sharma, Anjali; Liyanage, Wathsala; Tichý, Tomáš; Tenora, Lukáš; Su, Yu; Ha, Jisu; Hin, Niyada; Obayashi, Mizuho; Majer, Pavel; Kannan, Rangaramanujam M; Tsukamoto, Takashi; Ursini, Gianluca; Rais, Rana; Slusher, Barbara S; Zhu, Xiaolei

Mass spectrometry-guided discovery of novel GCPII inhibitor scaffolds

质谱引导下新型GCPII抑制剂骨架的发现

Wiseman, Robyn; Thomas, Ajit G; Janiszewski, John; Hoxie, Nate; Lee, Chae Bin; Wu, Ying; Tsukamoto, Takashi; Ye, Lin; Ronzetti, Michael; Shrimp, Jonathan H; Adderley, Davina; Rai, Ganesha; Rais, Rana; Alt, Jesse; Hall, Matthew D; Hu, Xin; Kales, Stephen C; Slusher, Barbara S

Neutral sphingomyelinase 2: A promising drug target for CNS disease

中性鞘磷脂酶2:中枢神经系统疾病的一种有前景的药物靶点

Huang, Meixiang; Stremlau, Matthew; Zavras, Jason; Zivko, Cristina; Thomas, Ajit G; Pietri, Peter; Machairaki, Vasiliki; Slusher, Barbara S

Recurrent Syncope in a 27-Year-Old Primigravida

一名27岁初产妇反复晕厥

Gavali, Vishal; Udyavar, Ameya; Desai, Ajit G; Mehta, Ashwin B

GCPII Inhibition Promotes Remyelination after Peripheral Nerve Injury in Aged Mice.

GCPII抑制剂可促进老年小鼠周围神经损伤后的髓鞘再生

Su Yu, Huang Meixiang, Thomas Ajit G, Maragakis John, Huizar Kaitlyn D J, Zheng Yuxin, Wu Ying, Farah Mohamed H, Slusher Barbara S

A gut-restricted glutamate carboxypeptidase II inhibitor reduces monocytic inflammation and improves preclinical colitis

肠道特异性谷氨酸羧肽酶II抑制剂可减轻单核细胞炎症并改善临床前结肠炎

Diane E Peters ,Lauren D Norris ,Lukáš Tenora ,Ivan Šnajdr ,András K Ponti ,Xiaolei Zhu ,Shinji Sakamoto ,Vijayabhaskar Veeravalli ,Manisha Pradhan ,Jesse Alt ,Ajit G Thomas ,Pavel Majer ,Rana Rais ,Christine McDonald ,Barbara S Slusher

Inhibiting tau-induced elevated nSMase2 activity and ceramides is therapeutic in an Alzheimer's disease mouse model

抑制 tau 诱导的 nSMase2 活性升高和神经酰胺对阿尔茨海默病小鼠模型具有治疗作用

Carolyn Tallon, Benjamin J Bell, Medhinee M Malvankar, Pragney Deme, Carlos Nogueras-Ortiz, Erden Eren, Ajit G Thomas, Kristen R Hollinger, Arindom Pal, Maja Mustapic, Meixiang Huang, Kaleem Coleman, Tawnjerae R Joe, Rana Rais, Norman J Haughey, Dimitrios Kapogiannis, Barbara S Slusher

Dendrimer-enabled targeted delivery attenuates glutamate excitotoxicity and improves motor function in a rabbit model of cerebral palsy

树枝状聚合物靶向递送可减轻脑瘫兔模型的谷氨酸兴奋毒性并改善运动功能

Fan Zhang, Zhi Zhang, Jesse Alt, Siva P Kambhampati, Anjali Sharma, Sarabdeep Singh, Elizabeth Nance, Ajit G Thomas, Camilo Rojas, Rana Rais, Barbara S Slusher, Rangaramanujam M Kannan, Sujatha Kannan

T cell metabolic reprogramming in acute kidney injury and protection by glutamine blockade

急性肾损伤中T细胞代谢重编程及谷氨酰胺阻断的保护作用

Kyungho Lee ,Elizabeth A Thompson ,Sepideh Gharaie ,Chirag H Patel ,Johanna T Kurzhagen ,Phillip M Pierorazio ,Lois J Arend ,Ajit G Thomas ,Sanjeev Noel ,Barbara S Slusher ,Hamid Rabb