日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Selective enhancement of the interneuron network and gamma-band power via GluN2C/GluN2D NMDA receptor potentiation

通过GluN2C/GluN2D NMDA受体增强选择性增强中间神经元网络和γ波段功率

Camp, Chad R; Banke, Tue G; Xing, Hao; Yu, Kuai; Perszyk, Riley E; Epplin, Matthew P; Akins, Nicholas S; Zhang, Jing; Benke, Tim A; Yuan, Hongjie; Liotta, Dennis C; Traynelis, Stephen F

Enhancement of hippocampal interneuron excitability by NMDA receptor positive allosteric modulation.

NMDA受体正向变构调节增强海马中间神经元兴奋性。

Xing Hao, Banke Tue G, Zhang Lu, Yu Kuai, Camp Chad R, Fritzemeier Russell G, Akins Nicholas S, Paladugu Srinu, Arcoria Paul J, Brady Brian R, Prikhodko Olga, Kennedy Matthew J, Liotta Dennis C, Yuan Hongjie, Traynelis Stephen F

Molecular mechanism of ligand gating and opening of NMDA receptor

NMDA受体配体门控和开放的分子机制

Chou, Tsung-Han; Epstein, Max; Fritzemeier, Russell G; Akins, Nicholas S; Paladugu, Srinu; Ullman, Elijah Z; Liotta, Dennis C; Traynelis, Stephen F; Furukawa, Hiro

Mechanisms of Action Underlying Conductance-Modifying Positive Allosteric Modulators of the NMDA Receptor.

NMDA受体电导调节正变构调节剂的作用机制

Ullman Elijah Z, Perszyk Riley E, Paladugu Srinu, Fritzemeier Russell G, Akins Nicholas S, Jacobs Leon, Liotta Dennis C, Traynelis Stephen F

Selective Enhancement of the Interneuron Network and Gamma-Band Power via GluN2C/GluN2D NMDA Receptor Potentiation

通过 GluN2C/GluN2D NMDA 受体增强选择性增强中间神经元网络和伽马波段功率

Camp, Chad R; Banke, Tue G; Xing, Hao; Yu, Kuai; Perszyk, Riley E; Epplin, Matthew P; Akins, Nicholas S; Zhang, Jing; Benke, Tim A; Yuan, Hongjie; Liotta, Dennis C; Traynelis, Stephen F

Novel GluN2B-Selective NMDA Receptor Negative Allosteric Modulator Possesses Intrinsic Analgesic Properties and Enhances Analgesia of Morphine in a Rodent Tail Flick Pain Model

一种新型的GluN2B选择性NMDA受体负变构调节剂具有内在镇痛特性,并能增强吗啡在啮齿动物甩尾痛模型中的镇痛作用。

Harris, Lynnea D; Regan, Michael C; Myers, Scott J; Nocilla, Kelsey A; Akins, Nicholas S; Tahirovic, Yesim A; Wilson, Lawrence J; Dingledine, Ray; Furukawa, Hiro; Traynelis, Stephen F; Liotta, Dennis C

Development of a Dihydroquinoline-Pyrazoline GluN2C/2D-Selective Negative Allosteric Modulator of the N-Methyl-d-aspartate Receptor

开发一种二氢喹啉-吡唑啉类GluN2C/2D选择性N-甲基-D-天冬氨酸受体负变构调节剂

D'Erasmo, Michael P; Akins, Nicholas S; Ma, Peipei; Jing, Yao; Swanger, Sharon A; Sharma, Savita K; Bartsch, Perry W; Menaldino, David S; Arcoria, Paul J; Bui, Thi-Thien; Pons-Bennaceur, Alexandre; Le, Phuong; Allen, James P; Ullman, Elijah Z; Nocilla, Kelsey A; Zhang, Jing; Perszyk, Riley E; Kim, Sukhan; Acker, Timothy M; Taz, Azmain; Burton, Samantha L; Coe, Kevin; Fritzemeier, Russell G; Burnashev, Nail; Yuan, Hongjie; Liotta, Dennis C; Traynelis, Stephen F

Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings

通过后期 Buchwald 偶联反应改善 ADME 特性的氨基杂环四氢异喹啉 CXCR4 拮抗剂

Nguyen, Huy H; Tahirovic, Yesim A; Truax, Valarie M; Wilson, Robert J; Jecs, Edgars; Miller, Eric J; Kim, Michelle B; Akins, Nicholas S; Xu, Lingjie; Jiang, Yi; Wang, Tao; Sum, Chi S; Cvijic, Mary E; Schroeder, Gretchen M; Wilson, Lawrence J; Liotta, Dennis C

Inhibition of Glycolysis and Glutaminolysis: An Emerging Drug Discovery Approach to Combat Cancer

抑制糖酵解和谷氨酰胺分解:一种对抗癌症的新兴药物发现方法

Akins, Nicholas S; Nielson, Tanner C; Le, Hoang V