日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Properties of Acute Activation and Inhibition of the β3 Homomeric GABA(A) Receptor Mediated by Protonation of Conserved Histidine Residues

β3同源GABA(A)受体急性激活和抑制的特性，由保守组氨酸残基的质子化介导

期刊:ACS Chemical Neuroscience
影响因子:3.9
doi:10.1021/acschemneuro.5c00256
Pierce, Spencer R; Germann, Allison L; Zhou, Yu; Menon, Saumith L; Gu, Xinghan; Lingle, Christopher J; Evers, Alex S; Steinbach, Joe Henry; Akk, Gustav
信号转导
发表日期：2025
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Null method to estimate the maximal PA at subsaturating concentrations of agonist

零假设法用于估算激动剂浓度低于饱和浓度时的最大PA值

期刊:Journal of General Physiology
影响因子:2.9
doi:10.1085/jgp.202413644
Germann, Allison L; Pierce, Spencer R; Steinbach, Joe Henry; Akk, Gustav
发表日期：2025
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Direct measurements of neurosteroid binding to specific sites on GABA(A) receptors

直接测量神经甾体与GABA(A)受体特定位点的结合情况

期刊:British Journal of Pharmacology
影响因子:7.7
doi:10.1111/bph.16490
Chintala, Satyanarayana M; Tateiwa, Hiroki; Qian, Mingxing; Xu, Yuanjian; Amtashar, Fatima; Chen, Zi-Wei; Kirkpatrick, Charles C; Bracamontes, John; Germann, Allison L; Akk, Gustav; Covey, Douglas F; Evers, Alex S
信号转导
发表日期：2024
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Tabernanthalog and ibogainalog inhibit the α7 and α9α10 nicotinic acetylcholine receptors via different mechanisms and with higher potency than the GABA(A) receptor and Ca(V)2.2 channel

Tabernanthalog 和 ibogainalog 通过不同的机制抑制 α7 和 α9α10 尼古丁乙酰胆碱受体，且其效力高于 GABA(A) 受体和 Ca(V)2.2 通道。

期刊:Biochemical Pharmacology
影响因子:5.6
doi:10.1016/j.bcp.2024.116183
Tae, Han-Shen; Ortells, Marcelo O; Yousuf, Arsalan; Xu, Sophia Q; Akk, Gustav; Adams, David J; Arias, Hugo R
信号转导
发表日期：2024
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Comparison of Behavioral Effects of GABAergic Low- and High-Efficacy Neuroactive Steroids in the Zebrafish Larvae Assay

斑马鱼幼体实验中低效和高效GABA能神经活性类固醇行为效应的比较

期刊:ACS Chemical Neuroscience
影响因子:3.9
doi:10.1021/acschemneuro.3c00836
Germann, Allison L; Xu, Yuanjian; Covey, Douglas F; Evers, Alex S; Akk, Gustav
发表日期：2024
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Stereospecific Properties and Intracellular Transport of Novel Intrinsically Fluorescent Neurosteroids.

新型固有荧光神经甾体的立体特异性及细胞内转运

期刊:ACS Chemical Neuroscience
影响因子:3.9
doi:10.1021/acschemneuro.4c00571
Akkerman Vibeke, Reinholdt Peter, Schnoor-Madsen Rasmus, Lauritsen Line, Bader Jad, Qian Minxing, Xu Yuanjiang, Akk Gustav, Scheidt Holger A, Müller Peter, Covey Douglas F, Evers Alex S, Kongsted Jacob, Wüstner Daniel
神经科学
细胞生物学
发表日期：2024
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Potentiation of the GABA(A)R reveals variable energetic contributions by etiocholanolone and propofol

GABA(A)R 的增强作用揭示了乙胆醇酮和丙泊酚的不同能量贡献。

期刊:Biophysical Journal
影响因子:3.1
doi:10.1016/j.bpj.2023.09.014
Pierce, Spencer R; Xu, Sophia Q; Germann, Allison L; Steinbach, Joe Henry; Akk, Gustav
发表日期：2024
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Inhibitory Actions of Potentiating Neuroactive Steroids in the Human α1β3γ2L γ-Aminobutyric Acid Type A Receptor

增强神经活性类固醇对人α1β3γ2L γ-氨基丁酸A型受体的抑制作用

期刊:Molecular Pharmacology
影响因子:3
doi:10.1124/molpharm.124.000960
Pierce, Spencer R; Germann, Allison L; Covey, Douglas F; Evers, Alex S; Steinbach, Joe Henry; Akk, Gustav
信号转导
Human
发表日期：2024
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The Mechanism of Enantioselective Neurosteroid Actions on GABA(A) Receptors

对映选择性神经甾体作用于GABA(A)受体的机制

期刊:Biomolecules
影响因子:4.8
doi:10.3390/biom13020341
Tateiwa, Hiroki; Chintala, Satyanarayana M; Chen, Ziwei; Wang, Lei; Amtashar, Fatima; Bracamontes, John; Germann, Allison L; Pierce, Spencer R; Covey, Douglas F; Akk, Gustav; Evers, Alex S
信号转导
发表日期：2023
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Perspective on the Relationship between GABAA Receptor Activity and the Apparent Potency of an Inhibitor

关于GABAA受体活性与抑制剂表观效力之间关系的观点

期刊:Current Neuropharmacology
影响因子:5.3
doi:10.2174/1570159X19666211104142433
Germann, Allison L; Pierce, Spencer R; Evers, Alex S; Steinbach, Joe Henry; Akk, Gustav
信号转导
表观遗传
发表日期：2022
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