Discovery of a novel 4-pyridyl SLC-0111 analog targeting tumor-associated carbonic anhydrase isoform IX through tail-based design approach with potent anticancer activity
通过基于尾部结构的设计方法,发现了一种靶向肿瘤相关碳酸酐酶IX同工酶的新型4-吡啶基SLC-0111类似物,该类似物具有强大的抗癌活性。
期刊:Frontiers in Chemistry
影响因子:4.2
doi:10.3389/fchem.2025.1571646
Hashem, Hamada; Abdelfattah, Shadwa; Hassan, Hesham M; Al-Emam, Ahmed; Alqarni, Mohammed; Alotaibi, Ghallab; Radwan, Ibrahim Taha; Kaur, Kirandeep; Rao, Devendra Pratap; Bräse, Stefan; Alkhammash, Abdullah