日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis, multi-target evaluation and DFT analysis of 6-hydroxychromone derived hydrazones with carbonic anhydrase I-II/acetylcholinesterase inhibition and antioxidant activity

6-羟基色酮衍生的腙类化合物的合成、多靶点评价及DFT分析及其碳酸酐酶I-II/乙酰胆碱酯酶抑制活性和抗氧化活性

Zareen, Wajeeha; Ahmed, Nadeem; Tokali, Feyzi Sinan; Islam, Talha; Al-Rashida, Mariya; Senol, Ayşe Merve; Ulucay, Orhan; Tawfeek, Ahmed Mohamed; Taslimi, Parham; Shafiq, Zahid; Islam, Mohammad Shahidul

Synthesis and biological evaluation of 6-hydroxychromone based thiosemicarbazones as potential antidiabetic and antioxidant agents

6-羟基色酮基硫代氨基脲类化合物的合成及生物学评价:作为潜在的抗糖尿病和抗氧化剂

Zareen, Wajeeha; Ahmed, Nadeem; Siddique, Farhan; Taslimi, Parham; Khan, Muhammad Ali; Islam, Talha; Ismail, Mostafa A; Al-Rashida, Mariya; Zaki, Magdi E A; Gomha, Sobhi M; Alharthy, Rima D; Shafiq, Zahid

Synthesis, in vitro, and in silico studies of 4-chlorophenyl-sulfonyl Indole based thiosemicarbazones as competitive α-glucosidase inhibitors

4-氯苯基磺酰基吲哚基硫代氨基脲类化合物作为竞争性α-葡萄糖苷酶抑制剂的合成、体外和计算机模拟研究

Naseer, Iqra; Ullah, Saeed; Batool, Zahra; Al-Rashida, Mariya; Islam, Talha; Khan, Ajmal; Hussain, Javid; Al-Harrasi, Ahmed; Shafiq, Zahid; Tawfeek, Ahmed Mohamed; Islam, Mohammad Shahidul

Design, synthesis, and multi-target evaluation of 4-phenyl quinoline-8-sulfonate thiosemicarbazones as potential anti-Alzheimer agents

4-苯基喹啉-8-磺酸硫代氨基脲类化合物的设计、合成及多靶点评价:作为潜在的抗阿尔茨海默病药物

Saeed, Rahma; Tariq, Hafiza Zara; Althobaiti, Aiysha; Sadeghian, Nastaran; Taslimi, Parham; Al-Rashida, Mariya; Islam, Talha; Thabet, Hamdy Khamees; Aftab, Hina; Şenol, Halil; Ameen, Mubashir; Li, Jing; Shafiq, Zahid

Sustainable approach for synthesis of new coumarin-linked Schiff bases in DABCO-based ionic liquid and their identification as aldose reductase inhibitors

在基于DABCO的离子液体中合成新型香豆素连接的席夫碱的可持续方法及其作为醛糖还原酶抑制剂的鉴定

Ishtiaq, Marium; Iqbal, Naved; Imran, Aqeel; Al-Rashida, Mariya; Rana, Sobia; Khan, Maria Aqeel; Iqbal, Jamshed; Hameed, Abdul

Synthesis, in vitro biological evaluation and in silico studies of novel pyrrolidine derived thiosemicarbazones as dihydrofolate reductase inhibitors

新型吡咯烷衍生的硫代氨基脲类化合物作为二氢叶酸还原酶抑制剂的合成、体外生物学评价和计算机模拟研究

Aftab, Hina; Ullah, Saeed; Khan, Ajmal; Al-Rashida, Mariya; Islam, Talha; Alshammari, Abdulrahman; Albekairi, Norah A; Taslimi, Parham; Al-Harrasi, Ahmed; Shafiq, Zahid; Alghamdi, Saeed

Optimization study and application of box-behnken model for probing eggshell supported transition metals based catalysts to synthesize hydrazone & dihydropyrimidinones

利用box-behnken模型优化研究并应用其在蛋壳负载过渡金属基催化剂合成腙和二氢嘧啶酮中的应用

Perveen, Rabia; Latif, Fiza; Abbas, Minahil; Ayub, Khurshid; Sarfaraz, Sehrish; Saeed, Muhammad; Rana, Sobia; Al-Rashida, Mariya; Nawaz, Muhammad Asif; Hameed, Abdul

Pyrazole derivatives of pyridine and naphthyridine as proapoptotic agents in cervical and breast cancer cells

吡啶和萘啶的吡唑衍生物作为宫颈癌和乳腺癌细胞的促凋亡剂

Rima D Alharthy, Faisal Rashid, Abida Ashraf, Zahid Shafiq, Steven Ford, Mariya Al-Rashida, Muhammad Yaqub, Jamshed Iqbal

Utilization of transition metal fluoride-based solid support catalysts for the synthesis of sulfonamides: carbonic anhydrase inhibitory activity and in silico study

利用过渡金属氟化物基固体载体催化剂合成磺酰胺:碳酸酐酶抑制活性及计算机模拟研究

Ali, Deedar; Amjad, Sayyeda Tayyeba; Shafique, Zainab; Naseer, Muhammad Moazzam; Al-Rashida, Mariya; Sindhu, Tayyaba Allamgir; Iftikhar, Shafia; Shah, Muhammad Raza; Hameed, Abdul; Iqbal, Jamshed

Synthesis, Carbonic Anhydrase II/IX/XII Inhibition, DFT, and Molecular Docking Studies of Hydrazide-Sulfonamide Hybrids of 4-Methylsalicyl- and Acyl-Substituted Hydrazide

4-甲基水杨酰基和酰基取代的酰肼-磺酰胺杂合物的合成、碳酸酐酶II/IX/XII抑制、DFT和分子对接研究

Khushal, Adil; Mumtaz, Amara; Shadoul, Wamda Ahmed; Zaidi, Syeda Huda Mehdi; Rafique, Hummera; Munir, Abida; Maalik, Aneela; Shah, Syed Jawad Ali; Baig, Ayesha; Khawaja, Wajiha; Al-Rashida, Mariya; Hashmi, Muhammad Ali; Iqbal, Jamshed