Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights
鉴定新的 4-(6-氧代吡嗪-1-基)苯磺酰胺作为针对碳酸酐酶、COX-2 和 5-LOX 酶的多靶点抗炎药物:合成、生物学评价和建模见解
期刊:Journal of Enzyme Inhibition and Medicinal Chemistry
影响因子:5.6
doi:10.1080/14756366.2023.2201407
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany