日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-based design of potent pyrazolo[1,5-a]pyrimidine CDK4/6 inhibitors: biological evaluation and computational validation

基于结构的强效吡唑并[1,5-a]嘧啶类CDK4/6抑制剂设计:生物学评价和计算验证

Binjubair, Faizah A; Elkotamy, Mahmoud S; Mattar, Amr A; Almutairy, Bjad K; Al-Rashood, Sara T; Eldesouki, Mohamed M; Bouajila, Jalloul; Abdel-Aziz, Hatem A; Fakhry, Mariam M

Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights

鉴定新的 4-(6-氧代吡嗪-1-基)苯磺酰胺作为针对碳酸酐酶、COX-2 和 5-LOX 酶的多靶点抗炎药物:合成、生物学评价和建模见解

Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany

Design and statistical optimisation of emulsomal nanoparticles for improved anti-SARS-CoV-2 activity of N-(5-nitrothiazol-2-yl)-carboxamido candidates: in vitro and in silico studies

乳化纳米粒子的设计和统计优化以提高 N-(5-硝基噻唑-2-基)-甲酰胺候选物的抗 SARS-CoV-2 活性:体外和计算机模拟研究

Ahmed A Al-Karmalawy, Dalia S El-Gamil, Rabeh El-Shesheny, Marwa Sharaky, Radwan Alnajjar, Omnia Kutkat, Yassmin Moatasim, Mohamed Elagawany, Sara T Al-Rashood, Faizah A Binjubair, Wagdy M Eldehna, Ayman M Noreddin, Mohamed Y Zakaria3

Synergistic Effect of Sophora japonica and Glycyrrhiza glabra Flavonoid-Rich Fractions on Wound Healing: In Vivo and Molecular Docking Studies

槐米和光果甘草富含黄酮类成分对伤口愈合的协同作用:体内和分子对接研究

Shaza H Aly, Ahmed M Elissawy, Abdulla M A Mahmoud, Fatma Sa'eed El-Tokhy, Sherif S Abdel Mageed, Hadia Almahli, Sara T Al-Rashood, Faizah A Binjubair, Mahmoud A El Hassab, Wagdy M Eldehna, Abd El-Nasser B Singab

Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activity

新型 3-(6-甲基吡啶-2-基)香豆素基查耳酮作为具有抗增殖活性的癌症相关碳酸酐酶 IX 和 XII 的选择性抑制剂

Haytham O Tawfik, Moataz A Shaldam, Alessio Nocentini, Rofaida Salem, Hadia Almahli, Sara T Al-Rashood, Claudiu T Supuran, Wagdy M Eldehna

2-Arylquinolines as novel anticancer agents with dual EGFR/FAK kinase inhibitory activity: synthesis, biological evaluation, and molecular modelling insights

2-芳基喹啉类化合物作为新型抗癌药物,具有双重EGFR/FAK激酶抑制活性:合成、生物学评价和分子建模研究

Elbadawi, Mostafa M; Eldehna, Wagdy M; Abd El-Hafeez, Amer Ali; Somaa, Warda R; Albohy, Amgad; Al-Rashood, Sara T; Agama, Keli K; Elkaeed, Eslam B; Ghosh, Pradipta; Pommier, Yves; Abe, Manabu

GC/MS analysis and potential synergistic effect of mandarin and marjoram oils on Helicobacter pylori

GC/MS分析及柑橘油和马郁兰油对幽门螺杆菌的潜在协同作用

Elkousy, Rawah H; Mostafa, Nada M; Abd-Alkhalek, Ahmed M; El Hassab, Mahmoud A; Al-Rashood, Sara T; Eldehna, Wagdy M; Eldahshan, Omayma A

Phytonutrients, Colorant Pigments, Phytochemicals, and Antioxidant Potential of Orphan Leafy Amaranthus Species

孤叶苋属植物的植物营养素、着色色素、植物化学物质和抗氧化潜力

Sarker, Umakanta; Rabbani, Md Golam; Oba, Shinya; Eldehna, Wagdy M; Al-Rashood, Sara T; Mostafa, Nada M; Eldahshan, Omayma A

In Silico Docking, Resistance Modulation and Biofilm Gene Expression in Multidrug-Resistant Acinetobacter baumannii via Cinnamic and Gallic Acids

肉桂酸和没食子酸对多重耐药鲍曼不动杆菌的计算机模拟对接、耐药性调节和生物膜基因表达的影响

Abdelaziz, Neveen A; Elkhatib, Walid F; Sherif, Mahmoud M; Abourehab, Mohammed A S; Al-Rashood, Sara T; Eldehna, Wagdy M; Mostafa, Nada M; Elleboudy, Nooran S

GC/MS Profiling, Anti-Collagenase, Anti-Elastase, Anti-Tyrosinase and Anti-Hyaluronidase Activities of a Stenocarpus sinuatus Leaves Extract

银叶树叶提取物的GC/MS分析、抗胶原酶、抗弹性蛋白酶、抗酪氨酸酶和抗透明质酸酶活性

Younis, Mai M; Ayoub, Iriny M; Mostafa, Nada M; El Hassab, Mahmoud A; Eldehna, Wagdy M; Al-Rashood, Sara T; Eldahshan, Omayma A