In Silico and in vitro evaluation of the anticancer effect of a 1,5-Benzodiazepin-2-One derivative (3b) revealing potent dual inhibition of HER2 and HDAC1.
通过计算机模拟和体外实验评估 1,5-苯并二氮杂卓-2-酮衍生物 (3b) 的抗癌作用,发现其对 HER2 和 HDAC1 具有强效的双重抑制作用
期刊:Scientific Reports
影响因子:3.9
doi:10.1038/s41598-025-97786-7
Al-Theyab Nada S, Bakheit Ahmad H, Lahmidi Sanae, Alanazi Mohammed Mufadhe, Ali Awadh M, Azzaoui Khalil, Essassi El Mokhtar, Mague Joel T, Hefnawy Mohamad, Alanazi Mohammed Mater, Alanazi Ashwag S