日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Preclinical characterization of [(18)F]T-008, a novel PET imaging radioligand for cholesterol 24-hydroxylase

[(18)F]T-008 是一种新型的胆固醇 24-羟化酶 PET 成像放射性配体,对其进行了临床前表征

Koike, Tatsuki; Constantinescu, Cristian C; Ikeda, Shuhei; Nishi, Toshiya; Sunahara, Eiji; Miyamoto, Maki; Cole, Patricia; Barret, Olivier; Alagille, David; Papin, Caroline; Morley, Thomas; Fowles, Krista; Seibyl, John; Tamagnan, Gilles; Kuroita, Takanobu

Dopamine D(1) Receptor Agonist PET Tracer Development: Assessment in Nonhuman Primates

多巴胺D(1)受体激动剂PET示踪剂的开发:在非人灵长类动物中的评估

Barret, Olivier; Zhang, Lei; Alagille, David; Constantinescu, Cristian C; Sandiego, Christine; Papin, Caroline; Sullivan, Jenna M; Morley, Thomas; Carroll, Vincent M; Seibyl, John; Chen, Jianqing; Lee, Chewah; Villalobos, Anabella; Gray, David; McCarthy, Timothy J; Tamagnan, Gilles

Intrastriatal alpha-synuclein fibrils in monkeys: spreading, imaging and neuropathological changes

猴子纹状体内 α-突触核蛋白原纤维:扩散、成像和神经病理学变化

Yaping Chu, Scott Muller, Adriana Tavares, Olivier Barret, David Alagille, John Seibyl, Gilles Tamagnan, Ken Marek, Kelvin C Luk, John Q Trojanowski, Virginia M Y Lee, Jeffrey H Kordower

T156. IN VIVO CHARACTERIZATION OF THE FIRST AGONIST DOPAMINE D1 RECEPTORS PET IMAGING TRACER [18F]MNI-968 IN HUMAN

T156. 首个多巴胺D1受体激动剂PET成像示踪剂[18F]MNI-968在人体内的体内表征

Hinderer, Christian; Katz, Nathan; Dyer, Cecilia; Goode, Tamara; Johansson, Julia; Bell, Peter; Richman, Laura; Buza, Elizabeth; Wilson, James M; Tamagnan, Gilles; Barret, Olivier; Alagille, David; Carroll, Vincent; Madonia, Jennifer; Constantinescu, Cristian; SanDiego, Christine; Papin, Caroline; Morley, Thomas; Russell, David; McCarthy, Timothy; Zhang, Lei; Gray, David; Villalobos, Anna; Lee, Chewah; Chen, Jianqing; Seibyl, John; Marek, Kenneth

Preclinical properties and human in vivo assessment of 123I-ABC577 as a novel SPECT agent for imaging amyloid-β

123I-ABC577 作为一种新型 SPECT 显像剂用于淀粉样β蛋白成像的临床前特性及人体体内评估

Maya, Yoshifumi; Okumura, Yuki; Kobayashi, Ryohei; Onishi, Takako; Shoyama, Yoshinari; Barret, Olivier; Alagille, David; Jennings, Danna; Marek, Kenneth; Seibyl, John; Tamagnan, Gilles; Tanaka, Akihiro; Shirakami, Yoshifumi

Comparison of [(11)C]TZ1964B and [(18)F]MNI659 for PET imaging brain PDE10A in nonhuman primates

比较 [(11)C]TZ1964B 和 [(18)F]MNI659 在非人灵长类动物脑 PDE10A PET 成像中的应用

Liu, Hui; Jin, Hongjun; Yue, Xuyi; Han, Junbin; Yang, Hao; Flores, Hubert; Su, Yi; Alagille, David; Perlmutter, Joel S; Tamagnan, Gilles; Tu, Zhude

Microfluidic continuous-flow radiosynthesis of [(18)F]FPEB suitable for human PET imaging

适用于人体PET成像的[(18)F]FPEB微流控连续流放射合成

Liang, Steven H; Yokell, Daniel L; Jackson, Raul N; Rice, Peter A; Callahan, Ronald; Johnson, Keith A; Alagille, David; Tamagnan, Gilles; Collier, Thomas Lee; Vasdev, Neil

Metabotropic glutamate receptor 5 antagonist protects dopaminergic and noradrenergic neurons from degeneration in MPTP-treated monkeys

代谢型谷氨酸受体 5 拮抗剂可保护接受 MPTP 治疗的猴子的多巴胺能和去甲肾上腺素能神经元免于退化

Gunasingh J Masilamoni, James W Bogenpohl, David Alagille, Kristen Delevich, Gilles Tamagnan, John R Votaw, Thomas Wichmann, Yoland Smith

Potent mGluR5 antagonists: pyridyl and thiazolyl-ethynyl-3,5-disubstituted-phenyl series

强效mGluR5拮抗剂:吡啶基和噻唑基乙炔基-3,5-二取代苯基系列

Alagille, David; DaCosta, Herve; Chen, Yelin; Hemstapat, Kamondanai; Rodriguez, Alice; Baldwin, Ronald M; Conn, P Jeffrey; Tamagnan, Gilles D

Synthesis and In Vitro Evaluation of Imidazo[1,2-b]pyridazines as Ligands for β-Amyloid Plaques

咪唑并[1,2-b]哒嗪类化合物作为β-淀粉样斑块配体的合成及体外评价

Zeng, Fanxing; Alagille, David; Tamagnan, Gilles D; Ciliax, Brian J; Levey, Allan I; Goodman, Mark M