Discovery of new 5-substituted-indole-2-carboxamides as dual epidermal growth factor receptor (EGFR)/cyclin dependent kinase-2 (CDK2) inhibitors with potent antiproliferative action
发现新型5-取代吲哚-2-甲酰胺类化合物作为双重表皮生长因子受体(EGFR)/细胞周期蛋白依赖性激酶-2(CDK2)抑制剂,具有强效抗增殖作用
期刊:RSC Medicinal Chemistry
影响因子:3.6
doi:10.1039/d3md00038a
Mohamed, Fatma A M; Alakilli, Saleha Y M; El Azab, Eman Fawzy; Baawad, Faris A M; Shaaban, Esraa Ibrahim A; Alrub, Heba Abu; Hendawy, Omnia; Gomaa, Hesham A M; Bakr, Adel G; Abdelrahman, Mostafa H; Trembleau, Laurent; Mohammed, Anber F; Youssif, Bahaa G M