Stepwise Structural Simplification of the Dihydroxyanthraquinone Moiety of a Multitarget Rhein-Based Anti-Alzheimer Lead to Improve Drug Metabolism and Pharmacokinetic Properties
逐步简化多靶点大黄酸类抗阿尔茨海默症药物二羟基蒽醌部分的结构以改善药物代谢和药代动力学特性
期刊:Pharmaceutics
影响因子:4.9
doi:10.3390/pharmaceutics16080982
Caterina Pont, Anna Sampietro, F Javier Pérez-Areales, Nunzia Cristiano, Agustí Albalat, Belén Pérez, Manuela Bartolini, Angela De Simone, Vincenza Andrisano, Marta Barenys, Elisabet Teixidó, Raimon Sabaté, M Isabel Loza, José Brea, Diego Muñoz-Torrero