日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of PXR Antagonist MI891 and PXR Degrader MI1013 and Their Roles in Hepatic Gene Regulation

PXR拮抗剂MI891和PXR降解剂MI1013的发现及其在肝脏基因调控中的作用

Rajamanikkam Kamaraj ,Ivana Mejdrová ,Maria Krutakova ,Tomas Smutny ,Kryštof Škach ,Klara Dohnalova ,Lucie Smutna ,Dharani Sai Sreekanth Nellore ,Jan Dusek ,Karel Chalupsky ,Jana Hricová ,Thales Kronenberger ,Aaron Stahl ,Markus Templin ,Albert Braeuning ,Radim Nencka ,Petr Pavek

Impact of perfluoroalkyl substances (PFAS) and PFAS mixtures on lipid metabolism in differentiated HepaRG cells as a model for human hepatocytes

全氟烷基物质 (PFAS) 和 PFAS 混合物对分化 HepaRG 细胞脂质代谢的影响(作为人类肝细胞的模型)

Faezeh Sadrabadi, Jimmy Alarcan, Heike Sprenger, Albert Braeuning, Thorsten Buhrke

In vitro screening of understudied PFAS with a focus on lipid metabolism disruption

对研究不足的 PFAS 进行体外筛选,重点关注脂质代谢紊乱

Lackson Kashobwe, Faezeh Sadrabadi, Albert Braeuning, Pim E G Leonards, Thorsten Buhrke, Timo Hamers

A multi-omics approach to elucidate okadaic acid-induced changes in human HepaRG hepatocarcinoma cells

采用多组学方法阐明冈田酸诱导的人类 HepaRG 肝癌细胞变化

Leonie T D Wuerger #, Heike Sprenger #, Ksenia Krasikova, Markus Templin, Aaron Stahl, Uta M Herfurth, Holger Sieg, Albert Braeuning

Structural Elucidation of Agrochemical Metabolic Transformation Products Based on Infrared Ion Spectroscopy to Improve In Silico Toxicity Assessment

基于红外离子光谱法对农用化学品代谢转化产物进行结构解析,以改进计算机毒性评估

Matthias J A Vink, Jimmy Alarcan, Jonathan Martens, Wybren Jan Buma, Albert Braeuning, Giel Berden, Jos Oomens

Pregnane X receptor activation remodels glucose metabolism to promote NAFLD development in obese mice

孕烷 X 受体激活重塑肥胖小鼠的葡萄糖代谢,促进 NAFLD 发展

Mikko Karpale, Outi Kummu, Olli Kärkkäinen, Marko Lehtonen, Juha Näpänkangas, Uta M Herfurth, Albert Braeuning, Jaana Rysä, Jukka Hakkola

Okadaic Acid Activates JAK/STAT Signaling to Affect Xenobiotic Metabolism in HepaRG Cells

冈田酸激活JAK/STAT信号传导影响HepaRG细胞中的外来化合物代谢

Leonie T D Wuerger, Felicia Kudiabor, Jimmy Alarcan, Markus Templin, Oliver Poetz, Holger Sieg, Albert Braeuning

Adverse outcome pathway-based analysis of liver steatosis in vitro using human liver cell lines

使用人类肝细胞系进行基于不良后果途径的体外肝脂肪变性分析

Mawien Karaca, Kristin Fritsche, Dajana Lichtenstein, Özlem Vural, Katrin Kreuzer, Jimmy Alarcan, Albert Braeuning, Philip Marx-Stoelting, Tewes Tralau

A human Caco-2-based co-culture model of the inflamed intestinal mucosa for particle toxicity studies

基于人类 Caco-2 的炎症肠粘膜共培养模型,用于颗粒毒性研究

Maxi B Paul, Marén Schlief, Hannes Daher, Albert Braeuning, Holger Sieg, Linda Böhmert

Analysis of hyperforin (St. John's wort) action at TRPC6 channel leads to the development of a new class of antidepressant drugs

分析金丝桃素(圣约翰草)对 TRPC6 通道的作用有助于开发一类新型抗抑郁药物

Yamina El Hamdaoui #, Fang Zheng #, Nikolas Fritz, Lian Ye, Mai Anh Tran, Kevin Schwickert, Tanja Schirmeister, Albert Braeuning, Dajana Lichtenstein, Ute A Hellmich, Dorothee Weikert, Markus Heinrich, Giulia Treccani, Michael K E Schäfer, Gabriel Nowak, Bernd Nürnberg, Christian Alzheimer, Christia