日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The synthetic triterpenoids CDDO-TFEA and CDDO-Me, but not CDDO, promote nuclear exclusion of BACH1 impairing its activity

合成三萜类化合物 CDDO-TFEA 和 CDDO-Me(而非 CDDO)可促进 BACH1 的核排斥,从而损害其活性

Laura Casares, Rita Moreno, Kevin X Ali, Maureen Higgins, Sharadha Dayalan Naidu, Graham Neill, Lena Cassin, Anders E Kiib, Esben B Svenningsen, Alberto Minassi, Tadashi Honda, Thomas B Poulsen, Clotilde Wiel, Volkan I Sayin, Albena T Dinkova-Kostova, David Olagnier, Laureano de la Vega

Curcumin-based-fluorescent probes targeting ALDH1A3 as a promising tool for glioblastoma precision surgery and early diagnosis

以 ALDH1A3 为靶点的姜黄素荧光探针有望成为胶质母细胞瘤精准手术和早期诊断的有力工具

Edoardo L M Gelardi #, Diego Caprioglio #, Giorgia Colombo, Erika Del Grosso, Daniele Mazzoletti, Daiana Mattoteia, Stefano Salamone, Davide M Ferraris, Eleonora Aronica, Giulia Nato, Annalisa Buffo, Menico Rizzi, Lorenzo Magrassi, Alberto Minassi, Silvia Garavaglia

Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex

吡唑-姜黄素通过破坏 CDK9/CyclinT1 复合物抑制心肌细胞肥大

Masafumi Funamoto, Yoichi Sunagawa, Mai Gempei, Kana Shimizu, Yasufumi Katanasaka, Satoshi Shimizu, Toshihide Hamabe-Horiike, Giovanni Appendino, Alberto Minassi, Andreas Koeberle, Maki Komiyama, Kiyoshi Mori, Koji Hasegawa, Tatsuya Morimoto

First thermostable CLIP- tag by rational design applied to an archaeal O6 -alkyl-guanine-DNA-alkyl-transferase

第一个经过合理设计的耐热 CLIP 标签应用于古细菌 O6-烷基鸟嘌呤-DNA-烷基转移酶

Rosa Merlo, Rosanna Mattossovich, Marianna Genta, Anna Valenti, Giovanni Di Mauro, Alberto Minassi, Riccardo Miggiano, Giuseppe Perugino

Identification of a Novel Curcumin Derivative Influencing Notch Pathway and DNA Damage as a Potential Therapeutic Agent in T-ALL

鉴定出一种影响 Notch 通路和 DNA 损伤的新型姜黄素衍生物作为 T-ALL 的潜在治疗剂

Nadezda Zhdanovskaya, Sara Lazzari, Diego Caprioglio, Mariarosaria Firrincieli, Chiara Maioli, Eleonora Pace, Daniela Imperio, Claudio Talora, Diana Bellavia, Saula Checquolo, Mattia Mori, Isabella Screpanti, Alberto Minassi, Rocco Palermo

Betulinic acid hydroxamate prevents colonic inflammation and fibrosis in murine models of inflammatory bowel disease

桦木酸羟肟酸酯可预防小鼠炎症性肠病模型中的结肠炎症和纤维化

María E Prados,Adela García-Martín,Juan D Unciti-Broceta,Belén Palomares ,Juan A Collado ,Alberto Minassi,Marco A Calzado ,Giovanni Appendino,Eduardo Muñoz

Betulinic Acid Hydroxamate is Neuroprotective and Induces Protein Phosphatase 2A-Dependent HIF-1α Stabilization and Post-transcriptional Dephosphorylation of Prolyl Hydrolase 2

桦木酸羟肟酸酯具有神经保护作用,并诱导蛋白磷酸酶 2A 依赖的 HIF-1α 稳定化和脯氨酰水解酶 2 的转录后去磷酸化

María E Prados #, Alejandro Correa-Sáez #, Juan D Unciti-Broceta, Martín Garrido-Rodríguez, Carla Jimenez-Jimenez, Massimiliano Mazzone, Alberto Minassi, Giovanni Appendino, Marco A Calzado, Eduardo Muñoz

The Oxidation of Phytocannabinoids to Cannabinoquinoids

植物大麻素氧化为大麻醌

Diego Caprioglio, Daiana Mattoteia, Federica Pollastro, Roberto Negri, Annalisa Lopatriello, Giuseppina Chianese, Alberto Minassi, Juan A Collado, Eduardo Munoz, Orazio Taglialatela-Scafati, Giovanni Appendino

The dimerization of Δ 9-tetrahydrocannabinolic acid A (THCA-A)

Δ9-四氢大麻酚酸A(THCA-A)的二聚化

Arben Cuadari, Federica Pollastro, Juan D Unciti-Broceta, Diego Caprioglio, Alberto Minassi, Annalisa Lopatriello, Eduardo Muñoz, Orazio Taglialatela-Scafati, Giovanni Appendino

Celecoxib inhibits proliferation and survival of chronic myelogeous leukemia (CML) cells via AMPK-dependent regulation of β-catenin and mTORC1/2

塞来昔布通过 AMPK 依赖性调节 β-catenin 和 mTORC1/2 来抑制慢性粒细胞白血病 (CML) 细胞的增殖和存活

Beatrice Riva, Marco De Dominici, Ilaria Gnemmi, Samanta A Mariani, Alberto Minassi, Valentina Minieri, Paolo Salomoni, Pier Luigi Canonico, Armando A Genazzani, Bruno Calabretta, Fabrizio Condorelli