日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, In Silico Studies and Inhibitory Activity towards Bcr-Abl, BTK and FLT3-ITD of New 2,6,9-Trisubstituted Purine Derivatives as Potential Agents for the Treatment of Leukaemia

新型 2,6,9-三取代嘌呤衍生物的设计、合成、计算机模拟研究以及对 Bcr-Abl、BTK 和 FLT3-ITD 的抑制活性,作为治疗白血病的潜在药物

Jeanluc Bertrand, Hana Dostálová, Vladimír Kryštof, Radek Jorda, Thalía Delgado, Alejandro Castro-Alvarez, Jaime Mella, David Cabezas, Mario Faúndez, Christian Espinosa-Bustos, Cristian O Salas

Synthesis, antitumor activity, 3D-QSAR and molecular docking studies of new iodinated 4-(3 H)-quinazolinones 3 N-substituted

新型碘化4-(3H)-喹唑啉酮3N-取代的合成、抗肿瘤活性、3D-QSAR和分子对接研究

Marcia Pérez-Fehrmann, Víctor Kesternich, Arturo Puelles, Víctor Quezada, Fernanda Salazar, Philippe Christen, Jonathan Castillo, Juan Guillermo Cárcamo, Alejandro Castro-Alvarez, Ronald Nelson

Substituted Purines as High-Affinity Histamine H3 Receptor Ligands

取代嘌呤作为高亲和力组胺 H3 受体配体

Christian Espinosa-Bustos, Luisa Leitzbach, Tito Añazco, María J Silva, Andrea Del Campo, Alejandro Castro-Alvarez, Holger Stark, Cristian O Salas