日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Repurposing Drugs as Bacteroides fragilis BFT-3 Inhibitors in the Animal Infection Model Galleria mellonella

在蜡螟动物感染模型中,将药物重新用于脆弱拟杆菌BFT-3抑制剂的治疗

Jiménez-Alesanco, Ana; Gómara-Lomero, Marta; Jeblaoui, Hajar; Vega, Sonia; Velázquez-Campoy, Adrián; Aínsa, José Antonio; Abián, Olga

Shedding Light on Dark Chemical Matter: The Discovery of a SARS-CoV-2 M(pro) Main Protease Inhibitor through Intensive Virtual Screening and In Vitro Evaluation

揭开暗化学物质的神秘面纱:通过密集虚拟筛选和体外评估发现SARS-CoV-2 M(pro)主蛋白酶抑制剂

Peralta-Moreno, Maria Nuria; Mena, Yago; Ortega-Alarcon, David; Jimenez-Alesanco, Ana; Vega, Sonia; Abian, Olga; Velazquez-Campoy, Adrian; Thomson, Timothy M; Pinto, Marta; Granadino-Roldán, José M; Santos Tomas, Maria; Perez, Juan J; Rubio-Martinez, Jaime

Development of an efficient NUPR1 inhibitor with anticancer activity

开发具有抗癌活性的有效 NUPR1 抑制剂

Xi Liu #, Ana Jimenez-Alesanco #, Zexian Li, Bruno Rizzuti, José L Neira, Matías Estaras, Ling Peng, Eduardo Chuluyan, Juan Garona, Florencia Gottardo, Adrián Velazquez-Campoy, Yi Xia, Olga Abian, Patricia Santofimia-Castaño, Juan Iovanna7

Ultrafast Metal-Free Microsupercapacitor Arrays Directly Store Instantaneous High-Voltage Electricity from Mechanical Energy Harvesters

超快无金属微型超级电容器阵列直接存储来自机械能收集器的瞬时高压电

Shiqian Chen, Zheng Li, Po-Han Huang, Virginia Ruiz, Yingchun Su, Yujie Fu, Yolanda Alesanco, B Gunnar Malm, Frank Niklaus, Jiantong Li

Repositioning small molecule drugs as allosteric inhibitors of the BFT-3 toxin from enterotoxigenic Bacteroides fragilis

将小分子药物重新定位为产肠毒素脆弱拟杆菌 BFT-3 毒素的变构抑制剂

Ana Jimenez-Alesanco, Ulrich Eckhard, Marta Asencio Del Rio, Sonia Vega, Tibisay Guevara, Adrian Velazquez-Campoy, Francesc Xavier Gomis-Rüth, Olga Abian

When Virtual Assistants Meet Teledermatology: Validation of a Virtual Assistant to Improve the Quality of Life of Psoriatic Patients

当虚拟助手遇上远程皮肤病学:验证虚拟助手在改善银屑病患者生活质量方面的有效性

Roca, Surya; Almenara, Manuel; Gilaberte, Yolanda; Gracia-Cazaña, Tamara; Morales Callaghan, Ana M; Murciano, Daniel; García, José; Alesanco, Álvaro

Enzyme/Nanocopper Hybrid Nanozymes: Modulating Enzyme-like Activity by the Protein Structure for Biosensing and Tumor Catalytic Therapy

酶/纳米铜杂化纳米酶:通过蛋白质结构调控酶样活性,用于生物传感和肿瘤催化治疗

Losada-Garcia, Noelia; Jimenez-Alesanco, Ana; Velazquez-Campoy, Adrian; Abian, Olga; Palomo, Jose M

Discovery of Diverse Natural Products as Inhibitors of SARS-CoV-2 Mpro Protease through Virtual Screening

通过虚拟筛选发现多种可作为 SARS-CoV-2 Mpro 蛋白酶抑制剂的天然产物

Jaime Rubio-Martínez, Ana Jiménez-Alesanco, Laura Ceballos-Laita, David Ortega-Alarcón, Sonia Vega, Cristina Calvo, Cristina Benítez, Olga Abian, Adrián Velázquez-Campoy, Timothy M Thomson, José Manuel Granadino-Roldán, Patricia Gómez-Gutiérrez, Juan J Pérez

Seleno-Functionalization of Quercetin Improves the Non-Covalent Inhibition of M(pro) and Its Antiviral Activity in Cells against SARS-CoV-2

槲皮素的硒化功能化可增强其对M(pro)的非共价抑制作用及其在细胞中对抗SARS-CoV-2的抗病毒活性。

Mangiavacchi, Francesca; Botwina, Pawel; Menichetti, Elena; Bagnoli, Luana; Rosati, Ornelio; Marini, Francesca; Fonseca, Sérgio F; Abenante, Laura; Alves, Diego; Dabrowska, Agnieszka; Kula-Pacurar, Anna; Ortega-Alarcon, David; Jimenez-Alesanco, Ana; Ceballos-Laita, Laura; Vega, Sonia; Rizzuti, Bruno; Abian, Olga; Lenardão, Eder J; Velazquez-Campoy, Adrian; Pyrc, Krzysztof; Sancineto, Luca; Santi, Claudio

Sub-Micromolar Inhibition of SARS-CoV-2 3CLpro by Natural Compounds

天然化合物对SARS-CoV-2 3CLpro的亚微摩尔级抑制作用

Rizzuti, Bruno; Ceballos-Laita, Laura; Ortega-Alarcon, David; Jimenez-Alesanco, Ana; Vega, Sonia; Grande, Fedora; Conforti, Filomena; Abian, Olga; Velazquez-Campoy, Adrian