日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Botanical Drug PBI-05204, a Supercritical CO2 Extract of Nerium Oleander, Is Synergistic With Radiotherapy in Models of Human Glioblastoma

植物药 PBI-05204 是夹竹桃的超临界 CO2 提取物,在人类胶质母细胞瘤模型中与放射疗法具有协同作用

Alessandro Colapietro, Peiying Yang, Alessandra Rossetti, Andrea Mancini, Flora Vitale, Sharmistha Chakraborty, Stefano Martellucci, Francesco Marampon, Vincenzo Mattei, Giovanni Luca Gravina, Roberto Iorio, Robert A Newman, Claudio Festuccia

Anticancer effects of ABTL0812, a clinical stage drug inducer of autophagy-mediated cancer cell death, in glioblastoma models

ABTL0812(一种临床阶段的自噬介导癌细胞死亡的药物诱导剂)在胶质母细胞瘤模型中的抗癌作用

Andrea Mancini, Alessandro Colapietro, Loredana Cristiano, Alessandra Rossetti, Vincenzo Mattei, Giovanni Luca Gravina, Héctor Perez-Montoyo, Marc Yeste-Velasco, Jose Alfon, Carles Domenech, Claudio Festuccia

ATX-101, a Peptide Targeting PCNA, Has Antitumor Efficacy Alone or in Combination with Radiotherapy in Murine Models of Human Glioblastoma

ATX-101 是一种靶向 PCNA 的肽,在人类胶质母细胞瘤小鼠模型中单独使用或与放射疗法联合使用均具有抗肿瘤功效

Giovanni Luca Gravina, Alessandro Colapietro, Andrea Mancini, Alessandra Rossetti, Stefano Martellucci, Luca Ventura, Martina Di Franco, Francesco Marampon, Vincenzo Mattei, Leda Assunta Biordi, Marit Otterlei, Claudio Festuccia

Multiple Antitumor Molecular Mechanisms Are Activated by a Fully Synthetic and Stabilized Pharmaceutical Product Delivering the Active Compound Sulforaphane (SFX-01) in Preclinical Model of Human Glioblastoma

在人类胶质母细胞瘤临床前模型中,一种完全合成且稳定的药物产品可激活多种抗肿瘤分子机制,提供活性化合物萝卜硫素 (SFX-01)

Alessandro Colapietro, Alessandra Rossetti, Andrea Mancini, Stefano Martellucci, Giuseppe Ocone, Fanny Pulcini, Leda Biordi, Loredana Cristiano, Vincenzo Mattei, Simona Delle Monache, Francesco Marampon, Giovanni Luca Gravina, Claudio Festuccia

The Botanical Drug PBI-05204, a Supercritical CO2 Extract of Nerium Oleander, Inhibits Growth of Human Glioblastoma, Reduces Akt/mTOR Activities, and Modulates GSC Cell-Renewal Properties

植物药 PBI-05204 是夹竹桃的超临界 CO2 提取物,可抑制人类胶质母细胞瘤的生长、降低 Akt/mTOR 活性并调节 GSC 细胞更新特性

Alessandro Colapietro, Peiying Yang, Alessandra Rossetti, Andrea Mancini, Flora Vitale, Stefano Martellucci, Tara L Conway, Sharmistha Chakraborty, Francesco Marampon, Vincenzo Mattei, Giovanni Luca Gravina, Assunta Leda Biordi, Daoyan Wei, Robert A Newman, Claudio Festuccia

Can the AGE/RAGE/ERK signalling pathway and the epithelial-to-mesenchymal transition interact in the pathogenesis of chronic rhinosinusitis with nasal polyps?

AGE/RAGE/ERK 信号通路和上皮-间质转化是否在慢性鼻窦炎伴鼻息肉的发病机制中相互作用?

Antonella Vetuschi, Simona Pompili, Gian Piero Di Marco, Federico Calvaruso, Enzo Iacomino, Lidia Angelosante, Claudio Festuccia, Alessandro Colapietro, Roberta Sferra

Antitumorigenic Effects of Inhibiting Ephrin Receptor Kinase Signaling by GLPG1790 against Colorectal Cancer Cell Lines In Vitro and In Vivo

GLPG1790 抑制 Ephrin 受体激酶信号对结直肠癌细胞系的体内外抗肿瘤作用

Alessandro Colapietro, Giovanni Luca Gravina, Francesco Petragnano, Irene Fasciani, Bianca Maria Scicchitano, Filip Beirinckx, Philippe Pujuguet, Laurent Saniere, Ellen Van der Aar, Daniela Musio, Francesca De Felice, Vincenzo Mattei, Stefano Martellucci, Roberto Maggio, Vincenzo Tombolini, Claudio

Dual CXCR4 and E-Selectin Inhibitor, GMI-1359, Shows Anti-Bone Metastatic Effects and Synergizes with Docetaxel in Prostate Cancer Cell Intraosseous Growth

CXCR4 和 E-选择素双重抑制剂 GMI-1359 具有抗骨转移作用,并与多西他赛协同作用促进前列腺癌细胞骨内生长

Claudio Festuccia, Andrea Mancini, Giovanni Luca Gravina, Alessandro Colapietro, Antonella Vetuschi, Simona Pompili, Luca Ventura, Simona Delle Monache, Roberto Iorio, Andrea Del Fattore, William Fogler, John Magnani

The Brain Penetrating and Dual TORC1/TORC2 Inhibitor, RES529, Elicits Anti-Glioma Activity and Enhances the Therapeutic Effects of Anti-Angiogenetic Compounds in Preclinical Murine Models

脑穿透性和双重 TORC1/TORC2 抑制剂 RES529 可引发抗胶质瘤活性并增强抗血管生成化合物在临床前小鼠模型中的治疗效果

Giovanni Luca Gravina, Andrea Mancini, Alessandro Colapietro, Simona Delle Monache, Roberta Sferra, Simona Pompili, Flora Vitale, Stefano Martellucci, Francesco Marampon, Vincenzo Mattei, Leda Biordi, David Sherris, Claudio Festuccia

The Small Molecule Ephrin Receptor Inhibitor, GLPG1790, Reduces Renewal Capabilities of Cancer Stem Cells, Showing Anti-Tumour Efficacy on Preclinical Glioblastoma Models

小分子 Ephrin 受体抑制剂 GLPG1790 可降低癌症干细胞的更新能力,在临床前胶质母细胞瘤模型上显示出抗肿瘤功效

Giovanni Luca Gravina, Andrea Mancini, Alessandro Colapietro, Simona Delle Monache, Roberta Sferra, Flora Vitale, Loredana Cristiano, Stefano Martellucci, Francesco Marampon, Vincenzo Mattei, Filip Beirinckx, Philippe Pujuguet, Laurent Saniere, Giocondo Lorenzon, Ellen van der Aar, Claudio Festuccia