日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BET N-terminal bromodomain inhibition selectively blocks Th17 cell differentiation and ameliorates colitis in mice

BET N 端溴结构域抑制选择性阻断 Th17 细胞分化并改善小鼠结肠炎

Kalung Cheung, Geming Lu, Rajal Sharma, Adam Vincek, Ruihua Zhang, Alexander N Plotnikov, Fan Zhang, Qiang Zhang, Ying Ju, Yuan Hu, Li Zhao, Xinye Han, Jamel Meslamani, Feihong Xu, Anbalagan Jaganathan, Tong Shen, Hongfa Zhu, Elena Rusinova, Lei Zeng, Jiachi Zhou, Jianjun Yang, Liang Peng, Michael O

Structure-guided design of potent diazobenzene inhibitors for the BET bromodomains

针对 BET 溴结构域的强效重氮苯抑制剂的结构引导设计

Guangtao Zhang, Alexander N Plotnikov, Elena Rusinova, Tong Shen, Keita Morohashi, Jennifer Joshua, Lei Zeng, Shiraz Mujtaba, Michael Ohlmeyer, Ming-Ming Zhou

Down-regulation of NF-κB transcriptional activity in HIV-associated kidney disease by BRD4 inhibition

BRD4 抑制可下调 HIV 相关肾脏疾病中的 NF-κB 转录活性

Guangtao Zhang, Ruijie Liu, Yifei Zhong, Alexander N Plotnikov, Weijia Zhang, Lei Zeng, Elena Rusinova, Guillermo Gerona-Nevarro, Natasha Moshkina, Jennifer Joshua, Peter Y Chuang, Michael Ohlmeyer, John Cijiang He, Ming-Ming Zhou

Structural basis of allele variation of human thiopurine-S-methyltransferase

人类硫嘌呤-S-甲基转移酶等位基因变异的结构基础

Hong Wu, John R Horton, Kevin Battaile, Abdellah Allali-Hassani, Fernando Martin, Hong Zeng, Peter Loppnau, Masoud Vedadi, Alexey Bochkarev, Alexander N Plotnikov, Xiaodong Cheng