A-loop interactions in Mer tyrosine kinase give rise to inhibitors with two-step mechanism and long residence time of binding
Mer 酪氨酸激酶中的 A-loop 相互作用产生具有两步机制和长结合停留时间的抑制剂
期刊:Biochemical Journal
影响因子:4.4
doi:10.1042/BCJ20200735
Alexander Pflug, Marianne Schimpl, J Willem M Nissink, Ross C Overman, Philip B Rawlins, Caroline Truman, Elizabeth Underwood, Juli Warwicker, Jon Winter-Holt, William McCoull