日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification and characterization of novel candidate compounds targeting 6- and 7-transmembrane μ-opioid receptor isoforms

针对 6 和 7 跨膜 μ-阿片受体异构体的新型候选化合物的鉴定和表征

Arjun Muralidharan, Alexander Samoshkin, Marino Convertino, Marjo Hannele Piltonen, Pavel Gris, Jian Wang, Changyu Jiang, Richard Klares 3rd, Alexander Linton, Ru-Rong Ji, William Maixner, Nikolay V Dokholyan, Jeffrey S Mogil, Luda Diatchenko

A functional substitution in the L-aromatic amino acid decarboxylase enzyme worsens somatic symptoms via a serotonergic pathway

L-芳香族氨基酸脱羧酶的功能性替代通过血清素途径加重躯体症状

Samar Khoury, Marjo H Piltonen, Anh-Tien Ton, Tiffany Cole, Alexander Samoshkin, Shad B Smith, Inna Belfer, Gary D Slade, Roger B Fillingim, Joel D Greenspan, Richard Ohrbach, William Maixner, G Gregory Neely, Adrian W R Serohijos, Luda Diatchenko

Stabilization of μ-opioid receptor facilitates its cellular translocation and signaling

μ-阿片受体的稳定有利于其细胞转位和信号传导

Cheng Zhu, Qingjian Han, Alexander Samoshkin, Marino Convertino, Alexander Linton, Edgar M Faison, Ru-Rong Ji, Luda Diatchenko, Nikolay V Dokholyan

Epiregulin and EGFR interactions are involved in pain processing

表皮调节素和 EGFR 相互作用参与疼痛处理

Loren J Martin, Shad B Smith, Arkady Khoutorsky, Claire A Magnussen, Alexander Samoshkin, Robert E Sorge, Chulmin Cho, Noosha Yosefpour, Sivaani Sivaselvachandran, Sarasa Tohyama, Tiffany Cole, Thang M Khuong, Ellen Mir, Dustin G Gibson, Jeffrey S Wieskopf, Susana G Sotocinal, Jean Sebastien Austin,

Structural and functional interactions between six-transmembrane μ-opioid receptors and β2-adrenoreceptors modulate opioid signaling

六跨膜 μ-阿片受体与 β2-肾上腺素受体之间的结构和功能相互作用调节阿片信号传导

Alexander Samoshkin, Marino Convertino, Chi T Viet, Jeffrey S Wieskopf, Oleg Kambur, Jaclyn Marcovitz, Pinkal Patel, Laura S Stone, Eija Kalso, Jeffrey S Mogil, Brian L Schmidt, William Maixner, Nikolay V Dokholyan, Luda Diatchenko

Differential expression of the alternatively spliced OPRM1 isoform μ-opioid receptor-1K in HIV-infected individuals

HIV 感染者中剪接的 OPRM1 异构体 μ-阿片受体-1K 的差异表达

Seth M Dever, Blair N Costin, Ruqiang Xu, Nazira El-Hage, Joyce Balinang, Alexander Samoshkin, Megan A O'Brien, Marypeace McRae, Luda Diatchenko, Pamela E Knapp, Kurt F Hauser

Human condensin function is essential for centromeric chromatin assembly and proper sister kinetochore orientation

人类凝聚蛋白功能对于着丝粒染色质组装和正确的姊妹动粒定位至关重要

Alexander Samoshkin, Alexei Arnaoutov, Lars E T Jansen, Ilia Ouspenski, Louis Dye, Tatiana Karpova, James McNally, Mary Dasso, Don W Cleveland, Alexander Strunnikov